Antonella Fais
A New Class of Benzo[b]thiophene-chalcones as Cholinesterase Inhibitors: Synthesis, Biological Evaluation, Molecular Docking and ADME Studies
2024-01-01 Delogu, GIOVANNA LUCIA; Begala, Michela; João Matos, Maria; Crucitti, Davide; Sogos, Valeria; Era, Benedetta; Fais, Antonella
Phytochemical Composition and Biological Activity
2024-01-01 Fais, A.; Era, B.
Advances in Sardinian Withania somnifera (L.) Dunal crops through phytochemical and biological approaches
2024-01-01 Maccioni, Delia; Falconieri, Danilo; Acquas, Elio; Kasture, Sanjay Bhaskar; Era, Benedetta; Fais, Antonella; Cocco, Emma; Maxia, Andrea
Exploring Asphodelus microcarpus as a source of xanthine oxidase inhibitors: Insights from in silico and in vitro studies
2024-01-01 DI PETRILLO, Amalia; Siguri, Chiara; Delogu, Giovanna L.; Fais, Antonella; Era, Benedetta; Floris, Sonia; Pintus, Francesca; Kumar, Amit; Fantini, MASSIMO CLAUDIO; Olla, Stefania
Template Entrance Channel as Possible Allosteric Inhibition and Resistance Site for Quinolines Tricyclic Derivatives in RNA Dependent RNA Polymerase of Bovine Viral Diarrhea Virus
2023-01-01 Srivastava, M.; Mittal, L.; Sarmadhikari, D.; Singh, V. K.; Fais, A.; Kumar, A.; Asthana, S.
Promising inhibition of diabetes-related enzymes and antioxidant properties of Ptilostemon casabonae leaves extract
2023-01-01 Sanna, Cinzia; Fais, Antonella; Era, Benedetta; Delogu, Giovanna L; Sanna, Enrico; Dazzi, Laura; Rosa, Antonella; Marengo, Arianna; Rubiolo, Patrizia; De Agostini, Antonio; Floris, Sonia; Pintus, Francesca
Design of 3-Phenylcoumarins and 3-Thienylcoumarins as Potent Xanthine Oxidase Inhibitors: Synthesis, Biological Evaluation, and Docking Studies
2023-01-01 Fais, A.; Pintus, F.; Era, B.; Floris, S.; Kumar, A.; Sarmadhikari, D.; Sogos, V.; Uriarte, E.; Asthana, S.; Matos, M. J.
Phytochemicals in structure-based drug discovery
2023-01-01 Kumar, A.; Baranwal, J.; Di Petrillo, A.; Floris, S.; Barse, B.; Fais, A.
Inhibitory Effect of Quercetin on Oxidative Endogen Enzymes: A Focus on Putative Binding Modes
2023-01-01 Olla, S.; Siguri, C.; Fais, A.; Era, B.; Fantini, M. C.; Di Petrillo, A.
Hydroxylated Coumarin-Based Thiosemicarbazones as Dual Antityrosinase and Antioxidant Agents
2023-01-01 Masuri, Sebastiano; Era, Benedetta; Pintus, Francesca; Cadoni, Enzo; Cabiddu, Maria Grazia; Fais, Antonella; Pivetta, Tiziana
Comparison of Different Green Extraction Techniques Used for the Extraction of Targeted Flavonoids from Edible Feijoa (Acca sellowiana (O.Berg) Burret) Flowers
2023-01-01 Gil, Katarzyna Angelika; Jokić, Stela; Cikoš, Ana-Marija; Banožić, Marija; Jakovljević Kovač, Martina; Fais, Antonella; Tuberoso, Carlo Ignazio Giovanni
Structural insight of new butyrylcholinesterase inhibitors based on benzylbenzofuran scaffold
2022-01-01 Delogu, Giovanna L.; Fais, Antonella; Pintus, Francesca; Goyal, Chinmayi; Matos, Maria J.; Era, Benedetta; Kumar, Amit
Hydroxy-3-Phenylcoumarins as Multitarget Compounds for Skin Aging Diseases: Synthesis, Molecular Docking and Tyrosinase, Elastase, Collagenase and Hyaluronidase Inhibition, and Sun Protection Factor
2022-01-01 Pintus, Francesca; Floris, Sonia; Fais, Antonella; Era, Benedetta; Kumar, Amit; Gatto, Gianluca; Uriarte, Eugenio; Matos, Maria João
Biopolymer: a sustainable material for food and medical applications
2022-01-01 Baranwal, Jaya; Barse, Brajesh; Fais, Antonella; Delogu, GIOVANNA LUCIA; Kumar, Amit
Euphorbia characias Extract: Inhibition of Skin Aging-Related Enzymes and Nanoformulation
2022-01-01 Pintus, F.; Floris, S.; Fais, A.; Era, B.; Porcedda, C.; Tuberoso, C. I. G.; Caddeo, C.
Quercetin and its derivates as antiviral potentials: A comprehensive review
2022-01-01 Di Petrillo, A.; Orru, G.; Fais, A.; Fantini, M. C.
Supercritical extraction of volatile and fixed oils from Petroselinum crispum L. seeds: chemical composition and biological activity
2022-01-01 Piras, A.; Porcedda, S.; Falconieri, D.; Fais, A.; Era, B.; Carta, G.; Rosa, A.
Design, Synthesis, and in Vitro Evaluation of 4-(4-Hydroxyphenyl)piperazine-Based Compounds Targeting Tyrosinase
2022-01-01 Mirabile, Salvatore; Paola Germanò, Maria; Fais, Antonella; Lombardo, Lisa; Ricci, Federico; Floris, Sonia; Cacciola, Anna; Rapisarda, Antonio; Gitto, Rosaria; Laura De Luca, And
Anti-aging potential of extracts from Washingtonia filifera seeds
2021-01-01 Era, B.; Floris, S.; Sogos, V.; Porcedda, C.; Piras, A.; Medda, R.; Fais, A.; Pintus, F.
Structural Characterisation and Assessment of the Novel Bacillus amyloliquefaciens RK3 Exopolysaccharide on the Improvement of Cognitive Function in Alzheimer’s Disease Mice
2021-01-01 Gangalla, Ravi; Gattu, Sampath; Palaniappan, Sivasankar; Ahamed, Maqusood; Macha, Baswaraju; Thampu, Raja Komuraiah; Fais, Antonella; Cincotti, Alberto; Gatto, Gianluca; Dama, Murali; Kumar, Amit
Evaluation of novel 4-(4-fluorobenzyl)piperazin-1-yl]-based compounds as competitive tyrosinase inhibitors endowed with anti-melanogenic effects
2021-01-01 Mirabile, Salvatore; Vittorio, Serena; Germanò, Maria Paola; Adornato, Ilenia; Ielo, Laura; Rapisarda, Antonio; Gitto, Rosaria; Pintus, Francesca; De Luca, Laura; Fais, Antonella
A new biological prospective for the 2-phenylbenzofurans as inhibitors of α-glucosidase and of the islet amyloid polypeptide formation
2021-01-01 Delogu, GIOVANNA LUCIA; Era, Benedetta; Floris, Sonia; Medda, Rosaria; Sogos, Valeria; Pintus, Francesca; Gatto, Gianluca; Kumar, Amit; Torstensdotter Westermark, Gunilla; Fais, Antonella
Washingtonia filifera seed extracts inhibit the islet amyloid polypeptide fibrils formations and α-amylase and α-glucosidase activity
2021-01-01 Floris, S.; Fais, A.; Medda, R.; Pintus, F.; Piras, A.; Kumar, A.; Kus, P. M.; Westermark, G. T.; Era, B.
Euphorbia characias: Phytochemistry and Biological Activities
2021-01-01 Fais, Antonella; Delogu, Giovanna Lucia; Floris, Sonia; Era, Benedetta; Medda, Rosaria; Pintus, Francesca
Looking for new xanthine oxidase inhibitors: 3-Phenylcoumarins versus 2-phenylbenzofurans
2020-01-01 Era, Benedetta; Delogu, Giovanna L.; Pintus, Francesca; Fais, Antonella; Gatto, Gianluca; Uriarte, Eugenio; Fernanda, Borges; Kumar, Amit; Matos, Maria J.
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety
2020-01-01 De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R.
4-Fluorobenzylpiperazine-containing derivatives as efficient inhibitors of mushroom tyrosinase
2020-01-01 Vittorio, Serena; Ielo, Laura; Mirabile, Salvatore; Gitto, Rosaria; Fais, Antonella; Floris, Sonia; Rapisarda, Antonio; Paola Germanò, Maria; De Luca, Laura
Substitution Effects on the Optoelectronic Properties of Coumarin Derivatives
2020-01-01 Kumar, Amit; Baccoli, Roberto; Fais, Antonella; Cincotti, Alberto; Pilia, Luca; Gatto, Gianluca
Supercritical CO2 Extraction of Waste Citrus Seeds: Chemical Composition, Nutritional and Biological Properties of Edible Fixed Oils
2019-01-01 Rosa, Antonella; Era, Benedetta; Masala, Carla; Nieddu, Mariella; Scano, Paola; Fais, Antonella; Porcedda, Silvia; Piras, Alessandra
Synthesis, molecular docking and cholinesterase inhibitory activity of hydroxylated 2-phenylbenzofuran derivatives
2019-01-01 Fais, Antonella; Kumar, Amit; Medda, Rosaria; Pintus, Francesca; Delogu, Francesco; Matos, Maria J.; Era, Benedetta; Delogu, Giovanna L.
Antibacterial Activity and Molecular Docking Studies of a Selected Series of Hydroxy-3-arylcoumarins
2019-01-01 Pisano, M. B.; Kumar, A.; Medda, R.; Gatto, G.; Pal, Rajesh; Fais, A.; Era, B.; Cosentino, S.; Uriarte, E.; Santana, L.; Pintus, F.; Matos, M. J.
Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile
2019-01-01 Ielo, L.; Deri, B.; Germanò, M. P.; Vittorio, S.; Mirabile, S.; Gitto, R.; Rapisarda, A.; Ronsisvalle, S.; Floris, S.; Pazy, Y.; Fais, A.; Fishman, A.; De, Luca
Chemical composition and enzyme inhibition of Phytolacca dioica L. seeds extracts
2019-01-01 DI PETRILLO, Amalia; María González-Paramás, Ana; Rosa, Antonella; Ruggiero, Valeria; Boylan, Fabio; Kumar, Amit; Pintus, Francesca; Santos-Buelga, Celestino; Fais, Antonella; Era, Benedetta
Phytochemical composition and the cholinesterase and xanthine oxidase inhibitory properties of seed extracts from the Washingtonia filifera palm fruit.
2019-01-01 Floris, Sonia; Fais, Antonella; Rosa, Antonella; Piras, Alessandra; Marzouki, Hanen; Medda, Rosaria; Gonz´alez-Paramas, Ana M.; Kumar, Amit; Santos-Buelga, Celestino; Era, Benedetta
Evaluation of antioxidant activities and chemical composition of Washingtonia filifera extracts.
2018-01-01 Floris, S.; Era, B.; Fais, A.; Porcedda, S.; Falconieri, D.; Rosa, A.; Marzouki, H.; Santos Buelga, C.; Piras, A.
Selected Enzyme Inhibitory Effects of Euphorbia characias Extracts
2018-01-01 Fais, Antonella; Era, Benedetta; Di Petrillo, Amalia; Floris, Sonia; Piano, Dario; Montoro, Paola; Tuberoso, Carlo Ignazio Giovanni; Medda, Rosaria; Pintus, Francesca
Novel 2-pheynlbenzofuran derivatives as selective butyrylcholinesterase inhibitors for Alzheimer’s disease
2018-01-01 Kumar, Amit; Pintus, Francesca; DI PETRILLO, Amalia; Medda, Rosaria; Caria, Paola; João Matos, Maria; Viña, Dolores; Pieroni, Enrico; Delogu, Francesco; Era, Benedetta; Delogu, Giovanna L.; Fais, Antonella
Sardinian honeys as sources of xanthine oxidase and tyrosinase inhibitors
2018-01-01 DI PETRILLO, Amalia; Santos-Buelga, Celestino; Era, Benedetta; González-Paramás, Ana Maria; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca; Fais, Antonella
Coumarin derivatives as promising xanthine oxidase inhibitors
2018-01-01 Fais, Antonella; Era, Benedetta; Asthana, Shailendra; Sogos, Valeria; Medda, Rosaria; Santana, Lourdes; Uriarte, Eugenio; João Matos, Maria; Delogu, Francesco; Kumar, Amit
Broad-range potential of Asphodelus microcarpus leaves extract for drug development
2017-01-01 DI PETRILLO, Amalia; Fais, Antonella; Pintus, Francesca; Santos Buelga, Celestino; Gonzalez Paramas, Ana M.; Piras, Vincenzo; Orru, Germano; Mameli, Antonello; Tramontano, Enzo; Frau, Aldo
New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies
2017-01-01 Pintus, Francesca; Matos, Maria J.; Vilar, Santiago; Hripcsak, George; Varela, Carla; Uriarte, Eugenio; Santana, Lourdes; Borges, Fernanda; Medda, Rosaria; DI PETRILLO, Amalia; Era, Benedetta; Fais, Antonella
Plasma phospholipase, γ-CEHC and antioxidant capacity in fibromyalgia
2017-01-01 Fais, Antonella; Cacace, Enrico; Atzori, Luigi; Era, Benedetta; Ruggiero, Valeria
Free amino acids in fibromyalgia syndrome: relationship with clinical picture
2017-01-01 Ruggiero, Valeria; Mura, Massimiliano; Cacace, Enrico; Era, Benedetta; Peri, Marcella; Sanna, Giuseppina; Fais, Antonella
Chemical composition of Lycium europaeum fruit oil obtained by supercritical CO2 extraction and evaluation of its antioxidant activity, cytotoxicity and cell absorption
2017-01-01 Rosa, Antonella; Maxia, Andrea; Putzu, Danilo; Atzeri, Angela; Era, Benedetta; Fais, Antonella; Sanna, Cinzia; Piras, Alessandra
Soluble adenosine deaminase activity in fibromyalgia syndrome
2016-01-01 Ruggiero, Valeria; Cacace, Enrico; Era, Benedetta; Fais, Antonella
2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: Synthesis, biological activity and molecular modeling
2016-01-01 Delogu, GIOVANNA LUCIA; Matos M., J; Fanti, M; Era, B; Medda, Rosaria; Pieroni, E; Fais, Antonella; Kumar, A; Pintus, Francesca
Synthesis and biological activity of 2-phenylbenzofuran derivatives as butyrylcholinerase inhibitors
2016-01-01 Delogu, Giovanna lucia; Pintus, Francesca; Fais, Antonella
Tyrosinase inhibition and antioxidant properties of Asphodelus microcarpus extracts
2016-01-01 DI PETRILLO, Amalia; González Paramás, Ana Maria; Era, Benedetta; Medda, Rosaria; Pintus, Francesca; Santos Buelga, Celestino; Fais, Antonella
Design and discovery of tyrosinase inhibitors based on a coumarin scaffold
2015-01-01 Matos, M. J.; Varela, C.; Vilar, S.; Hripcsak, G.; Borges, F.; Santana, L.; Uriarte, E.; Fais, Antonella; DI PETRILLO, Amalia; Pintus, Francesca; Era, Benedetta
Inhibitory effects of 3-heteroarylcoumarin derivatives on the activity of tyrosinase
2014-01-01 Di Petrillo, A; Fais, Antonella; Corda, M; Matos, Mj; B. Era, B.
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
A New Class of Benzo[b]thiophene-chalcones as Cholinesterase Inhibitors: Synthesis, Biological Evaluation, Molecular Docking and ADME Studies | 1-gen-2024 | Delogu, GIOVANNA LUCIA; Begala, Michela; João Matos, Maria; Crucitti, Davide; Sogos, Valeria; Era, Benedetta; Fais, Antonella | MOLECULES | - |
Phytochemical Composition and Biological Activity | 1-gen-2024 | Fais, A.; Era, B. | PLANTS | - |
Advances in Sardinian Withania somnifera (L.) Dunal crops through phytochemical and biological approaches | 1-gen-2024 | Maccioni, Delia; Falconieri, Danilo; Acquas, Elio; Kasture, Sanjay Bhaskar; Era, Benedetta; Fais, Antonella; Cocco, Emma; Maxia, Andrea | INDUSTRIAL CROPS AND PRODUCTS | - |
Exploring Asphodelus microcarpus as a source of xanthine oxidase inhibitors: Insights from in silico and in vitro studies | 1-gen-2024 | DI PETRILLO, Amalia; Siguri, Chiara; Delogu, Giovanna L.; Fais, Antonella; Era, Benedetta; Floris, Sonia; Pintus, Francesca; Kumar, Amit; Fantini, MASSIMO CLAUDIO; Olla, Stefania | CHEMICO-BIOLOGICAL INTERACTIONS | - |
Template Entrance Channel as Possible Allosteric Inhibition and Resistance Site for Quinolines Tricyclic Derivatives in RNA Dependent RNA Polymerase of Bovine Viral Diarrhea Virus | 1-gen-2023 | Srivastava, M.; Mittal, L.; Sarmadhikari, D.; Singh, V. K.; Fais, A.; Kumar, A.; Asthana, S. | PHARMACEUTICALS | - |
Promising inhibition of diabetes-related enzymes and antioxidant properties of Ptilostemon casabonae leaves extract | 1-gen-2023 | Sanna, Cinzia; Fais, Antonella; Era, Benedetta; Delogu, Giovanna L; Sanna, Enrico; Dazzi, Laura; Rosa, Antonella; Marengo, Arianna; Rubiolo, Patrizia; De Agostini, Antonio; Floris, Sonia; Pintus, Francesca | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Design of 3-Phenylcoumarins and 3-Thienylcoumarins as Potent Xanthine Oxidase Inhibitors: Synthesis, Biological Evaluation, and Docking Studies | 1-gen-2023 | Fais, A.; Pintus, F.; Era, B.; Floris, S.; Kumar, A.; Sarmadhikari, D.; Sogos, V.; Uriarte, E.; Asthana, S.; Matos, M. J. | CHEMMEDCHEM | - |
Phytochemicals in structure-based drug discovery | 1-gen-2023 | Kumar, A.; Baranwal, J.; Di Petrillo, A.; Floris, S.; Barse, B.; Fais, A. | - | Elsevier |
Inhibitory Effect of Quercetin on Oxidative Endogen Enzymes: A Focus on Putative Binding Modes | 1-gen-2023 | Olla, S.; Siguri, C.; Fais, A.; Era, B.; Fantini, M. C.; Di Petrillo, A. | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
Hydroxylated Coumarin-Based Thiosemicarbazones as Dual Antityrosinase and Antioxidant Agents | 1-gen-2023 | Masuri, Sebastiano; Era, Benedetta; Pintus, Francesca; Cadoni, Enzo; Cabiddu, Maria Grazia; Fais, Antonella; Pivetta, Tiziana | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
Comparison of Different Green Extraction Techniques Used for the Extraction of Targeted Flavonoids from Edible Feijoa (Acca sellowiana (O.Berg) Burret) Flowers | 1-gen-2023 | Gil, Katarzyna Angelika; Jokić, Stela; Cikoš, Ana-Marija; Banožić, Marija; Jakovljević Kovač, Martina; Fais, Antonella; Tuberoso, Carlo Ignazio Giovanni | PLANTS | - |
Structural insight of new butyrylcholinesterase inhibitors based on benzylbenzofuran scaffold | 1-gen-2022 | Delogu, Giovanna L.; Fais, Antonella; Pintus, Francesca; Goyal, Chinmayi; Matos, Maria J.; Era, Benedetta; Kumar, Amit | PHARMACEUTICALS | - |
Hydroxy-3-Phenylcoumarins as Multitarget Compounds for Skin Aging Diseases: Synthesis, Molecular Docking and Tyrosinase, Elastase, Collagenase and Hyaluronidase Inhibition, and Sun Protection Factor | 1-gen-2022 | Pintus, Francesca; Floris, Sonia; Fais, Antonella; Era, Benedetta; Kumar, Amit; Gatto, Gianluca; Uriarte, Eugenio; Matos, Maria João | MOLECULES | - |
Biopolymer: a sustainable material for food and medical applications | 1-gen-2022 | Baranwal, Jaya; Barse, Brajesh; Fais, Antonella; Delogu, GIOVANNA LUCIA; Kumar, Amit | POLYMERS | - |
Euphorbia characias Extract: Inhibition of Skin Aging-Related Enzymes and Nanoformulation | 1-gen-2022 | Pintus, F.; Floris, S.; Fais, A.; Era, B.; Porcedda, C.; Tuberoso, C. I. G.; Caddeo, C. | PLANTS | - |
Quercetin and its derivates as antiviral potentials: A comprehensive review | 1-gen-2022 | Di Petrillo, A.; Orru, G.; Fais, A.; Fantini, M. C. | PHYTOTHERAPY RESEARCH | - |
Supercritical extraction of volatile and fixed oils from Petroselinum crispum L. seeds: chemical composition and biological activity | 1-gen-2022 | Piras, A.; Porcedda, S.; Falconieri, D.; Fais, A.; Era, B.; Carta, G.; Rosa, A. | NATURAL PRODUCT RESEARCH | - |
Design, Synthesis, and in Vitro Evaluation of 4-(4-Hydroxyphenyl)piperazine-Based Compounds Targeting Tyrosinase | 1-gen-2022 | Mirabile, Salvatore; Paola Germanò, Maria; Fais, Antonella; Lombardo, Lisa; Ricci, Federico; Floris, Sonia; Cacciola, Anna; Rapisarda, Antonio; Gitto, Rosaria; Laura De Luca, And | CHEMMEDCHEM | - |
Anti-aging potential of extracts from Washingtonia filifera seeds | 1-gen-2021 | Era, B.; Floris, S.; Sogos, V.; Porcedda, C.; Piras, A.; Medda, R.; Fais, A.; Pintus, F. | PLANTS | - |
Structural Characterisation and Assessment of the Novel Bacillus amyloliquefaciens RK3 Exopolysaccharide on the Improvement of Cognitive Function in Alzheimer’s Disease Mice | 1-gen-2021 | Gangalla, Ravi; Gattu, Sampath; Palaniappan, Sivasankar; Ahamed, Maqusood; Macha, Baswaraju; Thampu, Raja Komuraiah; Fais, Antonella; Cincotti, Alberto; Gatto, Gianluca; Dama, Murali; Kumar, Amit | POLYMERS | - |
Evaluation of novel 4-(4-fluorobenzyl)piperazin-1-yl]-based compounds as competitive tyrosinase inhibitors endowed with anti-melanogenic effects | 1-gen-2021 | Mirabile, Salvatore; Vittorio, Serena; Germanò, Maria Paola; Adornato, Ilenia; Ielo, Laura; Rapisarda, Antonio; Gitto, Rosaria; Pintus, Francesca; De Luca, Laura; Fais, Antonella | CHEMMEDCHEM | - |
A new biological prospective for the 2-phenylbenzofurans as inhibitors of α-glucosidase and of the islet amyloid polypeptide formation | 1-gen-2021 | Delogu, GIOVANNA LUCIA; Era, Benedetta; Floris, Sonia; Medda, Rosaria; Sogos, Valeria; Pintus, Francesca; Gatto, Gianluca; Kumar, Amit; Torstensdotter Westermark, Gunilla; Fais, Antonella | INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES | - |
Washingtonia filifera seed extracts inhibit the islet amyloid polypeptide fibrils formations and α-amylase and α-glucosidase activity | 1-gen-2021 | Floris, S.; Fais, A.; Medda, R.; Pintus, F.; Piras, A.; Kumar, A.; Kus, P. M.; Westermark, G. T.; Era, B. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Euphorbia characias: Phytochemistry and Biological Activities | 1-gen-2021 | Fais, Antonella; Delogu, Giovanna Lucia; Floris, Sonia; Era, Benedetta; Medda, Rosaria; Pintus, Francesca | PLANTS | - |
Looking for new xanthine oxidase inhibitors: 3-Phenylcoumarins versus 2-phenylbenzofurans | 1-gen-2020 | Era, Benedetta; Delogu, Giovanna L.; Pintus, Francesca; Fais, Antonella; Gatto, Gianluca; Uriarte, Eugenio; Fernanda, Borges; Kumar, Amit; Matos, Maria J. | INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES | - |
Discovery of a new potent inhibitor of mushroom tyrosinase (Agaricus bisporus) containing 4-(4-hydroxyphenyl)piperazin-1-yl moiety | 1-gen-2020 | De Luca, L.; Germano, M. P.; Fais, A.; Pintus, F.; Buemi, M. R.; Vittorio, S.; Mirabile, S.; Rapisarda, A.; Gitto, R. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
4-Fluorobenzylpiperazine-containing derivatives as efficient inhibitors of mushroom tyrosinase | 1-gen-2020 | Vittorio, Serena; Ielo, Laura; Mirabile, Salvatore; Gitto, Rosaria; Fais, Antonella; Floris, Sonia; Rapisarda, Antonio; Paola Germanò, Maria; De Luca, Laura | CHEMMEDCHEM | - |
Substitution Effects on the Optoelectronic Properties of Coumarin Derivatives | 1-gen-2020 | Kumar, Amit; Baccoli, Roberto; Fais, Antonella; Cincotti, Alberto; Pilia, Luca; Gatto, Gianluca | APPLIED SCIENCES | - |
Supercritical CO2 Extraction of Waste Citrus Seeds: Chemical Composition, Nutritional and Biological Properties of Edible Fixed Oils | 1-gen-2019 | Rosa, Antonella; Era, Benedetta; Masala, Carla; Nieddu, Mariella; Scano, Paola; Fais, Antonella; Porcedda, Silvia; Piras, Alessandra | EUROPEAN JOURNAL OF LIPID SCIENCE AND TECHNOLOGY | - |
Synthesis, molecular docking and cholinesterase inhibitory activity of hydroxylated 2-phenylbenzofuran derivatives | 1-gen-2019 | Fais, Antonella; Kumar, Amit; Medda, Rosaria; Pintus, Francesca; Delogu, Francesco; Matos, Maria J.; Era, Benedetta; Delogu, Giovanna L. | BIOORGANIC CHEMISTRY | - |
Antibacterial Activity and Molecular Docking Studies of a Selected Series of Hydroxy-3-arylcoumarins | 1-gen-2019 | Pisano, M. B.; Kumar, A.; Medda, R.; Gatto, G.; Pal, Rajesh; Fais, A.; Era, B.; Cosentino, S.; Uriarte, E.; Santana, L.; Pintus, F.; Matos, M. J. | MOLECULES | - |
Exploiting the 1-(4-fluorobenzyl)piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and biological profile | 1-gen-2019 | Ielo, L.; Deri, B.; Germanò, M. P.; Vittorio, S.; Mirabile, S.; Gitto, R.; Rapisarda, A.; Ronsisvalle, S.; Floris, S.; Pazy, Y.; Fais, A.; Fishman, A.; De, Luca | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Chemical composition and enzyme inhibition of Phytolacca dioica L. seeds extracts | 1-gen-2019 | DI PETRILLO, Amalia; María González-Paramás, Ana; Rosa, Antonella; Ruggiero, Valeria; Boylan, Fabio; Kumar, Amit; Pintus, Francesca; Santos-Buelga, Celestino; Fais, Antonella; Era, Benedetta | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Phytochemical composition and the cholinesterase and xanthine oxidase inhibitory properties of seed extracts from the Washingtonia filifera palm fruit. | 1-gen-2019 | Floris, Sonia; Fais, Antonella; Rosa, Antonella; Piras, Alessandra; Marzouki, Hanen; Medda, Rosaria; Gonz´alez-Paramas, Ana M.; Kumar, Amit; Santos-Buelga, Celestino; Era, Benedetta | RSC ADVANCES | - |
Evaluation of antioxidant activities and chemical composition of Washingtonia filifera extracts. | 1-gen-2018 | Floris, S.; Era, B.; Fais, A.; Porcedda, S.; Falconieri, D.; Rosa, A.; Marzouki, H.; Santos Buelga, C.; Piras, A. | - | - |
Selected Enzyme Inhibitory Effects of Euphorbia characias Extracts | 1-gen-2018 | Fais, Antonella; Era, Benedetta; Di Petrillo, Amalia; Floris, Sonia; Piano, Dario; Montoro, Paola; Tuberoso, Carlo Ignazio Giovanni; Medda, Rosaria; Pintus, Francesca | BIOMED RESEARCH INTERNATIONAL | - |
Novel 2-pheynlbenzofuran derivatives as selective butyrylcholinesterase inhibitors for Alzheimer’s disease | 1-gen-2018 | Kumar, Amit; Pintus, Francesca; DI PETRILLO, Amalia; Medda, Rosaria; Caria, Paola; João Matos, Maria; Viña, Dolores; Pieroni, Enrico; Delogu, Francesco; Era, Benedetta; Delogu, Giovanna L.; Fais, Antonella | SCIENTIFIC REPORTS | - |
Sardinian honeys as sources of xanthine oxidase and tyrosinase inhibitors | 1-gen-2018 | DI PETRILLO, Amalia; Santos-Buelga, Celestino; Era, Benedetta; González-Paramás, Ana Maria; Tuberoso, CARLO IGNAZIO GIOVANNI; Medda, Rosaria; Pintus, Francesca; Fais, Antonella | FOOD SCIENCE AND BIOTECHNOLOGY | - |
Coumarin derivatives as promising xanthine oxidase inhibitors | 1-gen-2018 | Fais, Antonella; Era, Benedetta; Asthana, Shailendra; Sogos, Valeria; Medda, Rosaria; Santana, Lourdes; Uriarte, Eugenio; João Matos, Maria; Delogu, Francesco; Kumar, Amit | INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES | - |
Broad-range potential of Asphodelus microcarpus leaves extract for drug development | 1-gen-2017 | DI PETRILLO, Amalia; Fais, Antonella; Pintus, Francesca; Santos Buelga, Celestino; Gonzalez Paramas, Ana M.; Piras, Vincenzo; Orru, Germano; Mameli, Antonello; Tramontano, Enzo; Frau, Aldo | BMC MICROBIOLOGY | - |
New insights into highly potent tyrosinase inhibitors based on 3-heteroarylcoumarins: Anti-melanogenesis and antioxidant activities, and computational molecular modeling studies | 1-gen-2017 | Pintus, Francesca; Matos, Maria J.; Vilar, Santiago; Hripcsak, George; Varela, Carla; Uriarte, Eugenio; Santana, Lourdes; Borges, Fernanda; Medda, Rosaria; DI PETRILLO, Amalia; Era, Benedetta; Fais, Antonella | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Plasma phospholipase, γ-CEHC and antioxidant capacity in fibromyalgia | 1-gen-2017 | Fais, Antonella; Cacace, Enrico; Atzori, Luigi; Era, Benedetta; Ruggiero, Valeria | INTERNATIONAL JOURNAL OF RHEUMATIC DISEASES | - |
Free amino acids in fibromyalgia syndrome: relationship with clinical picture | 1-gen-2017 | Ruggiero, Valeria; Mura, Massimiliano; Cacace, Enrico; Era, Benedetta; Peri, Marcella; Sanna, Giuseppina; Fais, Antonella | SCANDINAVIAN JOURNAL OF CLINICAL & LABORATORY INVESTIGATION | - |
Chemical composition of Lycium europaeum fruit oil obtained by supercritical CO2 extraction and evaluation of its antioxidant activity, cytotoxicity and cell absorption | 1-gen-2017 | Rosa, Antonella; Maxia, Andrea; Putzu, Danilo; Atzeri, Angela; Era, Benedetta; Fais, Antonella; Sanna, Cinzia; Piras, Alessandra | FOOD CHEMISTRY | - |
Soluble adenosine deaminase activity in fibromyalgia syndrome | 1-gen-2016 | Ruggiero, Valeria; Cacace, Enrico; Era, Benedetta; Fais, Antonella | JOURNAL OF MUSCULOSKELETAL PAIN | - |
2-Phenylbenzofuran derivatives as butyrylcholinesterase inhibitors: Synthesis, biological activity and molecular modeling | 1-gen-2016 | Delogu, GIOVANNA LUCIA; Matos M., J; Fanti, M; Era, B; Medda, Rosaria; Pieroni, E; Fais, Antonella; Kumar, A; Pintus, Francesca | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Synthesis and biological activity of 2-phenylbenzofuran derivatives as butyrylcholinerase inhibitors | 1-gen-2016 | Delogu, Giovanna lucia; Pintus, Francesca; Fais, Antonella | - | MDPI |
Tyrosinase inhibition and antioxidant properties of Asphodelus microcarpus extracts | 1-gen-2016 | DI PETRILLO, Amalia; González Paramás, Ana Maria; Era, Benedetta; Medda, Rosaria; Pintus, Francesca; Santos Buelga, Celestino; Fais, Antonella | BMC COMPLEMENTARY AND ALTERNATIVE MEDICINE | - |
Design and discovery of tyrosinase inhibitors based on a coumarin scaffold | 1-gen-2015 | Matos, M. J.; Varela, C.; Vilar, S.; Hripcsak, G.; Borges, F.; Santana, L.; Uriarte, E.; Fais, Antonella; DI PETRILLO, Amalia; Pintus, Francesca; Era, Benedetta | RSC ADVANCES | - |
Inhibitory effects of 3-heteroarylcoumarin derivatives on the activity of tyrosinase | 1-gen-2014 | Di Petrillo, A; Fais, Antonella; Corda, M; Matos, Mj; B. Era, B. | - | - |
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