Filippo Cottiglia
Limonoids from Melia azeradach fruits as inhibitors of Flaviviruses
In corso di stampa Sanna, Giuseppina; Madeddu, S; Giliberti, G; La Colla, P; Cottiglia, Filippo; Ntali, N; Caboni, Pierluigi
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPβ phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea
2024-01-01 Huang, Shiu-Wen; Hsu, Ming Jen; Chen, Hsiu-Chen; Meleddu, Rita; Distinto, Simona; Maccioni, Elias; Cottiglia, Filippo
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms
2023-01-01 Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, Andrea; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action
2023-01-01 Corona, A.; Meleddu, R.; Delelis, O.; Subra, F.; Cottiglia, F.; Esposito, F.; Distinto, S.; Maccioni, E.; Tramontano, E.
Effects of docosanyl ferulate, a constituent of Withania somnifera, on ethanol- and morphine-elicited conditioned place preference and ERK phosphorylation in the accumbens shell of CD1 mice
2022-01-01 Maccioni, R.; Serra, M.; Marongiu, J.; Cottiglia, F.; Maccioni, E.; Bassareo, V.; Morelli, M.; Kasture, S. B.; Acquas, E.
Formulation and In Vitro Efficacy Assessment of Teucrium marum Extract Loading Hyalurosomes Enriched with Tween 80 and Glycerol
2022-01-01 Firoznezhad, M.; Castangia, I.; Tuberoso, C. I. G.; Cottiglia, F.; Marongiu, F.; Porceddu, M.; Usach, I.; Escribano-Ferrer, E.; Manca, M. L.; Manconi, M.
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions
2021-01-01 Meleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Mátyus, Péter; Maccioni, Elias
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function
2021-01-01 Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives
2021-01-01 Meleddu, R.; Deplano, S.; Maccioni, E.; Ortuso, F.; Cottiglia, F.; Secci, D.; Onali, A.; Sanna, E.; Angeli, A.; Angius, R.; Alcaro, S.; Supuran, C. T.; Distinto, S.
The biologically active compound of Withania somnifera (L.) Dunal, docosanyl ferulate, is endowed with potent anxiolytic properties but devoid of typical benzodiazepine-like side effects
2021-01-01 Maccioni, R.; Cottiglia, F.; Maccioni, E.; Talani, G.; Sanna, E.; Bassareo, V.; Kasture, S. B.; Acquas, E.
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII
2020-01-01 Meleddu, R.; Distinto, S.; Cottiglia, F.; Angius, R.; Caboni, P.; Angeli, A.; Melis, C.; Deplano, S.; Alcaro, S.; Ortuso, F.; Supuran, C. T.; Maccioni, E.
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation
2020-01-01 Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F.
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases
2019-01-01 Distinto, S.; Meleddu, R.; Ortuso, F.; Cottiglia, F.; Deplano, S.; SOUSA SEQUEIRA, ANA LISA; Melis, C.; Fois, B.; Angeli, A.; Capasso, C.; Angius, Riccardo; Alcaro, S.; Supuran, C. T.; Maccioni, E.
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators
2019-01-01 Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACCHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids
2019-01-01 Meleddu, Rita; Petrikaite, Vilma; Distinto, Simona; Arridu, Antonella; Angius, Rossella; Serusi, Lorenzo; Škarnulytė, Laura; Endriulaitytė, Ugnė; Paškevičiu̅tė, Miglė; Cottiglia, Filippo; Gaspari, Marco; Taverna, Domenico; Deplano, Serenella; Fois, Benedetta; Maccioni, Elias
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors
2018-01-01 Melis, Claudia; Distinto, Simona; Bianco, Giulia; Meleddu, Rita; Cottiglia, Filippo; Fois, Benedetta; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Maccioni, Elias
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides
2018-01-01 Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Gaspari, Marco; Taverna, Domenico; Melis, Claudia; Angeli, Andrea; Bianco, Giulia; Deplano, Serenella; Fois, Benedetta; Del Prete, Sonia; Capasso, Clemente; Alcaro, Stefano; Ortuso, Francesco; Yanez, Matilde; Supuran Claudiu, T.; Maccioni, Elias
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders
2017-01-01 Fois, Benedetta; Bianco, Giulia; Sonar, Vijay P.; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Melis, Claudia; Marras, Luisa; Pompei, Raffaello; Floris, Costantino; Caboni, Pierluigi; Cottiglia, Filippo
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action
2017-01-01 Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms
2017-01-01 Bianco, Giulia; Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Gaspari, Marco; Melis, Claudia; Corona, Angela; Angius, Rossella; Angeli, Andrea; Taverna, Domenico; Alcaro, Stefano; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T.; Maccioni, Elias
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B
2017-01-01 Meleddu, Rita; Distinto, Simona; Cirilli, Roberto; Alcaro, Stefano; Yanez, Matilde; Sanna, MARIA LUISA; Corona, Angela; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Maccioni, Elias
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase
2017-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia; Cottiglia, Filippo; Maccioni, Elias
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors
2017-01-01 Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clemente; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, Elias
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase
2017-01-01 Sonar, VIJAY PRAKASH; Corona, Angela; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Fois, Benedetta; Floris, Costantino; Malpure, Nilesh V.; Alcaro, Stefano; Tramontano, Enzo; Cottiglia, Filippo
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold
2016-01-01 Distinto, Simona; Meleddu, Rita; Yanez, Matilde; Cirilli, Roberto; Bianco, Giulia; Sanna, MARIA LUISA; Arridu, Antonella; Cossu, Pietro; Cottiglia, Filippo; Faggi, Cristina; Ortuso, Francesco; Alcaro, Stefano; Maccioni, Elias
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida
2016-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Maccioni, Elias; Arridu, Antonella; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Sanna, Adriana; DE LOGU, Alessandro
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase
2015-01-01 Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias
Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies
2015-01-01 Ruiu, S; Anzani, N; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Alcaro, S; Maccioni, Elias; Distinto, Simona; Cottiglia, Filippo
Limonoids from Melia azedarach fruits as inhibitors of flaviviruses and mycobacterium tubercolosis
2015-01-01 Sanna, Giuseppina; Madeddu, Silvia; Giliberti, Gabriele; Ntalli, Nikoletta G.; Cottiglia, Filippo; DE LOGU, Alessandro; Agus, Emanuela; Caboni, Pierluigi
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII
2015-01-01 Meleddu, Rita; Maccioni, Elias; Distinto, Simona; Bianco, Giulia; Melis, Claudia; Alcaro, Stefano; Cottiglia, Filippo; Ceruso, Mariangela; Supuran, Claudiu T.
Withania somnifera root extract prolongs analgesia and suppresses hyperalgesia in mice treated with morphine
2014-01-01 Orrù, A; Marchese, G; Casu, G; Casu, Ma; Kasture, S; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACHINO; Mascia, Mp; Anzani, Nicola; Ruiu, S.
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase
2014-01-01 Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, C; Esposito, Francesca; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Artese, A; Scalise, D; Fresta, M; Arridu, A; Ortuso, F; Maccioni, Elias; Tramontano, Enzo
Withania somnifera prevents acquisition and expression of morphine-elicited conditioned place preference
2013-01-01 Ruiu, S; Longoni, Rosanna; Spina, Liliana; Orru', Alessandro; Cottiglia, Filippo; Collu, Maria; Kasture, S; Acquas, ELIO MARIA GIOACHINO
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors
2013-01-01 Ruiu, S; Anzani, Nicola; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S; Cottiglia, Filippo
Cytotoxic phloroglucinols from the leaves of Myrtus communis
2012-01-01 Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina
Lumichrome and Phenyllactic Acid as Chemical Markers of Thistle (Galactites tomentosa Moench) Honey
2011-01-01 Tuberoso, CARLO IGNAZIO GIOVANNI; Bifulco, Ersilia; Caboni, Pierluigi; Sarais, Giorgia; Cottiglia, Filippo; Floris, I.
Ungeremine effectively targets mammalian as well as bacterial type I and type II topoisomerases
2011-01-01 Casu, Laura; Cottiglia, Filippo; Leonti, Marco; DE LOGU, Alessandro; Agus, E; Tse Dinh, Yc; Lombardo, V; Sissi, C.
Benzophenones from the root of the Popoluca Amerindian plant Securidaca diversifolia
2010-01-01 Casu, Laura; Cottiglia, Filippo; Pompei, Raffaello; Leonti, Marco
Falcarinol is a covalent cannabinoid CB1 receptor antagonist and induces pro-allergic effects in skin
2010-01-01 Leonti, Marco; Casu, Laura; Raduner, S; Cottiglia, Filippo; Floris, Costantino; ALTMANN K., H; Gertsch, J.
Floral markers of strawberry tree (Arbutus unedo L.) honey
2010-01-01 Tuberoso, CARLO IGNAZIO GIOVANNI; Bifulco, Ersilia; Caboni, Pierluigi; Cottiglia, Filippo; Cabras, P; Floris, I.
A pterocarpan from the seeds of Bituminaria morisiana
2010-01-01 Leonti, Marco; Casu, Laura; Gertsch, J; Bonsignore, L; Floris, Costantino; Casu, Mariano; Cottiglia, Filippo
A chromone from Seseli praecox (Apiaceae)
2010-01-01 Leonti, Marco; Casu, Laura; SOLINAS M., N; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Gertsch, J; Saba, A. R.
Cytotoxic tirucallane triterpenoids from Melia azedarach fruits
2010-01-01 Ntalli, Nikoletta; Cottiglia, Filippo; Bueno, Ca; Alché, Le; Leonti, Marco; Vargiu, S; Bifulco, Ersilia; MENKISSOGLU SPIROUDI, U; Caboni, Pierluigi
Benzophenones from the roots of the Popoluca Amerindian medicinal plant Securidaca diversifolia (L.) S.F. Blake
2010-01-01 Casu, Laura; Solinas, Mn; Saba, Ar; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Laconi, S; Pompei, Raffaello; Leonti, Marco
Bioactivity guided and random isolation of polyacetylenic compounds from Seseli praecox
2009-01-01 Leonti, Marco; Gertsch, J; Casu, Laura; Cottiglia, Filippo; SOLINAS M., N; Bonsignore, L; Raduner, S; Altmann, K. H.
New cytotoxic saturated and unsaturated cyclohexanones from Anthemis maritima
2008-01-01 Collu, F; Bonsignore, L; Casu, Mariano; Floris, Costantino; Gertschcjurg, ; Cottiglia, Filippo
Antiherpevirus activity of Artemisia arborescens essential oil and inhibition of lateral diffusion in Vero cells
2007-01-01 Saddi, M; Sanna, Adriana; Cottiglia, Filippo; Chisu, L; Casu, Laura; Bonsignore, L; DE LOGU, Alessandro
Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: Extraction, biological analysis, and computational study
2006-01-01 Chimenti, F; Cottiglia, Filippo; Bonsignore, L; Casu, Laura; Casu, Mariano; Floris, Costantino; Secci, D; Bolasco, A; Cimenti, P; Granese, A; Befani, O; Turini, P; Alcano, S; Ortuso, F; Trombetta, G; Loizzo, A; Guarino, I.
Cytotoxic diacetylenic spiroketalenol ethers from Plagius flosculosus
2006-01-01 Casu, Laura; Bonsignore, L; Pinna, M; Casu, Mariano; Floris, Costantino; Gertsch, J; Cottiglia, Filippo
New cytotoxic prenylated isoflavonoids from Bituminaria morisiana
2005-01-01 Cottiglia, Filippo; Casu, Laura; L., Bonsignore; Casu, Mariano; Floris, Costantino; Leonti, Marco; J., Gertsch; J., Heilmann
Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
---|---|---|---|---|
Limonoids from Melia azeradach fruits as inhibitors of Flaviviruses | In corso di stampa | Sanna, Giuseppina; Madeddu, S; Giliberti, G; La Colla, P; Cottiglia, Filippo; Ntali, N; Caboni, Pierluigi | ANTIVIRAL RESEARCH | - |
Suppression of lipopolysaccharide-induced COX-2 expression via p38MAPK, JNK, and C/EBPβ phosphorylation inhibition by furomagydarin A, a benzofuran glycoside from Magydaris pastinacea | 1-gen-2024 | Huang, Shiu-Wen; Hsu, Ming Jen; Chen, Hsiu-Chen; Meleddu, Rita; Distinto, Simona; Maccioni, Elias; Cottiglia, Filippo | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms | 1-gen-2023 | Sequeira, Lisa; Distinto, Simona; Meleddu, Rita; Gaspari, Marco; Angeli, Andrea; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Borges, Fernanda; Uriarte, Eugenio; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
5-Nitro-3-(2-(4-phenylthiazol-2-yl)hydrazineylidene)indolin-2-one derivatives inhibit HIV-1 replication by a multitarget mechanism of action | 1-gen-2023 | Corona, A.; Meleddu, R.; Delelis, O.; Subra, F.; Cottiglia, F.; Esposito, F.; Distinto, S.; Maccioni, E.; Tramontano, E. | FRONTIERS IN CELLULAR AND INFECTION MICROBIOLOGY | - |
Effects of docosanyl ferulate, a constituent of Withania somnifera, on ethanol- and morphine-elicited conditioned place preference and ERK phosphorylation in the accumbens shell of CD1 mice | 1-gen-2022 | Maccioni, R.; Serra, M.; Marongiu, J.; Cottiglia, F.; Maccioni, E.; Bassareo, V.; Morelli, M.; Kasture, S. B.; Acquas, E. | PSYCHOPHARMACOLOGY | - |
Formulation and In Vitro Efficacy Assessment of Teucrium marum Extract Loading Hyalurosomes Enriched with Tween 80 and Glycerol | 1-gen-2022 | Firoznezhad, M.; Castangia, I.; Tuberoso, C. I. G.; Cottiglia, F.; Marongiu, F.; Porceddu, M.; Usach, I.; Escribano-Ferrer, E.; Manca, M. L.; Manconi, M. | NANOMATERIALS | - |
Exploring new scaffolds for the dual inhibition of HIV-1 RT polymerase and ribonuclease associated functions | 1-gen-2021 | Meleddu, Rita; Corona, Angela; Distinto, Simona; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Secci, Daniela; Onali, Alessia; Sanna, Erica; Esposito, Francesca; Cirone, Italo; Ortuso, Francesco; Alcaro, Stefano; Tramontano, Enzo; Mátyus, Péter; Maccioni, Elias | MOLECULES | - |
Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function | 1-gen-2021 | Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives | 1-gen-2021 | Meleddu, R.; Deplano, S.; Maccioni, E.; Ortuso, F.; Cottiglia, F.; Secci, D.; Onali, A.; Sanna, E.; Angeli, A.; Angius, R.; Alcaro, S.; Supuran, C. T.; Distinto, S. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
The biologically active compound of Withania somnifera (L.) Dunal, docosanyl ferulate, is endowed with potent anxiolytic properties but devoid of typical benzodiazepine-like side effects | 1-gen-2021 | Maccioni, R.; Cottiglia, F.; Maccioni, E.; Talani, G.; Sanna, E.; Bassareo, V.; Kasture, S. B.; Acquas, E. | JOURNAL OF PSYCHOPHARMACOLOGY | - |
New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII | 1-gen-2020 | Meleddu, R.; Distinto, S.; Cottiglia, F.; Angius, R.; Caboni, P.; Angeli, A.; Melis, C.; Deplano, S.; Alcaro, S.; Ortuso, F.; Supuran, C. T.; Maccioni, E. | ACS MEDICINAL CHEMISTRY LETTERS | - |
Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation | 1-gen-2020 | Fois, B.; Distinto, S.; Meleddu, R.; Deplano, S.; Maccioni, E.; Floris, C.; Rosa, A.; Nieddu, M.; Caboni, P.; Sissi, C.; Angeli, A.; Supuran, C. T.; Cottiglia, F. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases | 1-gen-2019 | Distinto, S.; Meleddu, R.; Ortuso, F.; Cottiglia, F.; Deplano, S.; SOUSA SEQUEIRA, ANA LISA; Melis, C.; Fois, B.; Angeli, A.; Capasso, C.; Angius, Riccardo; Alcaro, S.; Supuran, C. T.; Maccioni, E. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators | 1-gen-2019 | Sonar, Vijay P.; Fois, Benedetta; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACCHINO; Kasture, Sanjay; Floris, Costantino; Colombo, Daniele; Sissi, Claudia; Sanna, Enrico; Talani, Giuseppe | JOURNAL OF NATURAL PRODUCTS | - |
Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids | 1-gen-2019 | Meleddu, Rita; Petrikaite, Vilma; Distinto, Simona; Arridu, Antonella; Angius, Rossella; Serusi, Lorenzo; Škarnulytė, Laura; Endriulaitytė, Ugnė; Paškevičiu̅tė, Miglė; Cottiglia, Filippo; Gaspari, Marco; Taverna, Domenico; Deplano, Serenella; Fois, Benedetta; Maccioni, Elias | ACS MEDICINAL CHEMISTRY LETTERS | - |
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors | 1-gen-2018 | Melis, Claudia; Distinto, Simona; Bianco, Giulia; Meleddu, Rita; Cottiglia, Filippo; Fois, Benedetta; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Maccioni, Elias | ACS MEDICINAL CHEMISTRY LETTERS | - |
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides | 1-gen-2018 | Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Gaspari, Marco; Taverna, Domenico; Melis, Claudia; Angeli, Andrea; Bianco, Giulia; Deplano, Serenella; Fois, Benedetta; Del Prete, Sonia; Capasso, Clemente; Alcaro, Stefano; Ortuso, Francesco; Yanez, Matilde; Supuran Claudiu, T.; Maccioni, Elias | ACS MEDICINAL CHEMISTRY LETTERS | - |
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders | 1-gen-2017 | Fois, Benedetta; Bianco, Giulia; Sonar, Vijay P.; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Melis, Claudia; Marras, Luisa; Pompei, Raffaello; Floris, Costantino; Caboni, Pierluigi; Cottiglia, Filippo | JOURNAL OF NATURAL PRODUCTS | - |
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action | 1-gen-2017 | Esposito, Francesca; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; Distinto, Simona; Corona, Angela; Lianza, Mariacaterina; Piano, Dario; Tacchini, Massimo; Maccioni, Elias; Cottiglia, Filippo; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; Tramontano, Enzo | PATHOGENS AND DISEASE | - |
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms | 1-gen-2017 | Bianco, Giulia; Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Gaspari, Marco; Melis, Claudia; Corona, Angela; Angius, Rossella; Angeli, Andrea; Taverna, Domenico; Alcaro, Stefano; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T.; Maccioni, Elias | ACS MEDICINAL CHEMISTRY LETTERS | - |
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B | 1-gen-2017 | Meleddu, Rita; Distinto, Simona; Cirilli, Roberto; Alcaro, Stefano; Yanez, Matilde; Sanna, MARIA LUISA; Corona, Angela; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Maccioni, Elias | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2017 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia; Cottiglia, Filippo; Maccioni, Elias | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors | 1-gen-2017 | Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clemente; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, Elias | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2017 | Sonar, VIJAY PRAKASH; Corona, Angela; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Fois, Benedetta; Floris, Costantino; Malpure, Nilesh V.; Alcaro, Stefano; Tramontano, Enzo; Cottiglia, Filippo | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold | 1-gen-2016 | Distinto, Simona; Meleddu, Rita; Yanez, Matilde; Cirilli, Roberto; Bianco, Giulia; Sanna, MARIA LUISA; Arridu, Antonella; Cossu, Pietro; Cottiglia, Filippo; Faggi, Cristina; Ortuso, Francesco; Alcaro, Stefano; Maccioni, Elias | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida | 1-gen-2016 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Maccioni, Elias; Arridu, Antonella; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Sanna, Adriana; DE LOGU, Alessandro | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2015 | Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Francesca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, Elias | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies | 1-gen-2015 | Ruiu, S; Anzani, N; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Alcaro, S; Maccioni, Elias; Distinto, Simona; Cottiglia, Filippo | JOURNAL OF NATURAL PRODUCTS | - |
Limonoids from Melia azedarach fruits as inhibitors of flaviviruses and mycobacterium tubercolosis | 1-gen-2015 | Sanna, Giuseppina; Madeddu, Silvia; Giliberti, Gabriele; Ntalli, Nikoletta G.; Cottiglia, Filippo; DE LOGU, Alessandro; Agus, Emanuela; Caboni, Pierluigi | PLOS ONE | - |
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII | 1-gen-2015 | Meleddu, Rita; Maccioni, Elias; Distinto, Simona; Bianco, Giulia; Melis, Claudia; Alcaro, Stefano; Cottiglia, Filippo; Ceruso, Mariangela; Supuran, Claudiu T. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Withania somnifera root extract prolongs analgesia and suppresses hyperalgesia in mice treated with morphine | 1-gen-2014 | Orrù, A; Marchese, G; Casu, G; Casu, Ma; Kasture, S; Cottiglia, Filippo; Acquas, ELIO MARIA GIOACHINO; Mascia, Mp; Anzani, Nicola; Ruiu, S. | PHYTOMEDICINE | - |
Design, synthesis, and biological evaluation of 1,3-diarylpropenones as dual inhibitors of HIV-1 reverse transcriptase | 1-gen-2014 | Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, C; Esposito, Francesca; Bianco, G; Corona, Angela; Cottiglia, Filippo; Alcaro, S; Parolin, C; Artese, A; Scalise, D; Fresta, M; Arridu, A; Ortuso, F; Maccioni, Elias; Tramontano, Enzo | CHEMMEDCHEM | - |
Withania somnifera prevents acquisition and expression of morphine-elicited conditioned place preference | 1-gen-2013 | Ruiu, S; Longoni, Rosanna; Spina, Liliana; Orru', Alessandro; Cottiglia, Filippo; Collu, Maria; Kasture, S; Acquas, ELIO MARIA GIOACHINO | BEHAVIOURAL PHARMACOLOGY | - |
N-Alkyl dien- and trienamides from the roots of Otanthus maritimus with binding affinity for opioid and cannabinoid receptors | 1-gen-2013 | Ruiu, S; Anzani, Nicola; Orrù, A; Floris, Costantino; Caboni, Pierluigi; Maccioni, Elias; Distinto, Simona; Alcaro, S; Cottiglia, Filippo | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Cytotoxic phloroglucinols from the leaves of Myrtus communis | 1-gen-2012 | Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina | JOURNAL OF NATURAL PRODUCTS | - |
Lumichrome and Phenyllactic Acid as Chemical Markers of Thistle (Galactites tomentosa Moench) Honey | 1-gen-2011 | Tuberoso, CARLO IGNAZIO GIOVANNI; Bifulco, Ersilia; Caboni, Pierluigi; Sarais, Giorgia; Cottiglia, Filippo; Floris, I. | JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | - |
Ungeremine effectively targets mammalian as well as bacterial type I and type II topoisomerases | 1-gen-2011 | Casu, Laura; Cottiglia, Filippo; Leonti, Marco; DE LOGU, Alessandro; Agus, E; Tse Dinh, Yc; Lombardo, V; Sissi, C. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Benzophenones from the root of the Popoluca Amerindian plant Securidaca diversifolia | 1-gen-2010 | Casu, Laura; Cottiglia, Filippo; Pompei, Raffaello; Leonti, Marco | PHYTOCHEMISTRY LETTERS | - |
Falcarinol is a covalent cannabinoid CB1 receptor antagonist and induces pro-allergic effects in skin | 1-gen-2010 | Leonti, Marco; Casu, Laura; Raduner, S; Cottiglia, Filippo; Floris, Costantino; ALTMANN K., H; Gertsch, J. | BIOCHEMICAL PHARMACOLOGY | - |
Floral markers of strawberry tree (Arbutus unedo L.) honey | 1-gen-2010 | Tuberoso, CARLO IGNAZIO GIOVANNI; Bifulco, Ersilia; Caboni, Pierluigi; Cottiglia, Filippo; Cabras, P; Floris, I. | JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | - |
A pterocarpan from the seeds of Bituminaria morisiana | 1-gen-2010 | Leonti, Marco; Casu, Laura; Gertsch, J; Bonsignore, L; Floris, Costantino; Casu, Mariano; Cottiglia, Filippo | NATURAL MEDICINES | - |
A chromone from Seseli praecox (Apiaceae) | 1-gen-2010 | Leonti, Marco; Casu, Laura; SOLINAS M., N; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Gertsch, J; Saba, A. R. | NATURAL PRODUCT COMMUNICATIONS | - |
Cytotoxic tirucallane triterpenoids from Melia azedarach fruits | 1-gen-2010 | Ntalli, Nikoletta; Cottiglia, Filippo; Bueno, Ca; Alché, Le; Leonti, Marco; Vargiu, S; Bifulco, Ersilia; MENKISSOGLU SPIROUDI, U; Caboni, Pierluigi | MOLECULES | - |
Benzophenones from the roots of the Popoluca Amerindian medicinal plant Securidaca diversifolia (L.) S.F. Blake | 1-gen-2010 | Casu, Laura; Solinas, Mn; Saba, Ar; Cottiglia, Filippo; Caboni, Pierluigi; Floris, Costantino; Laconi, S; Pompei, Raffaello; Leonti, Marco | PHYTOCHEMISTRY LETTERS | - |
Bioactivity guided and random isolation of polyacetylenic compounds from Seseli praecox | 1-gen-2009 | Leonti, Marco; Gertsch, J; Casu, Laura; Cottiglia, Filippo; SOLINAS M., N; Bonsignore, L; Raduner, S; Altmann, K. H. | - | - |
New cytotoxic saturated and unsaturated cyclohexanones from Anthemis maritima | 1-gen-2008 | Collu, F; Bonsignore, L; Casu, Mariano; Floris, Costantino; Gertschcjurg, ; Cottiglia, Filippo | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Antiherpevirus activity of Artemisia arborescens essential oil and inhibition of lateral diffusion in Vero cells | 1-gen-2007 | Saddi, M; Sanna, Adriana; Cottiglia, Filippo; Chisu, L; Casu, Laura; Bonsignore, L; DE LOGU, Alessandro | ANNALS OF CLINICAL MICROBIOLOGY AND ANTIMICROBIALS | - |
Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: Extraction, biological analysis, and computational study | 1-gen-2006 | Chimenti, F; Cottiglia, Filippo; Bonsignore, L; Casu, Laura; Casu, Mariano; Floris, Costantino; Secci, D; Bolasco, A; Cimenti, P; Granese, A; Befani, O; Turini, P; Alcano, S; Ortuso, F; Trombetta, G; Loizzo, A; Guarino, I. | JOURNAL OF NATURAL PRODUCTS | - |
Cytotoxic diacetylenic spiroketalenol ethers from Plagius flosculosus | 1-gen-2006 | Casu, Laura; Bonsignore, L; Pinna, M; Casu, Mariano; Floris, Costantino; Gertsch, J; Cottiglia, Filippo | JOURNAL OF NATURAL PRODUCTS | - |
New cytotoxic prenylated isoflavonoids from Bituminaria morisiana | 1-gen-2005 | Cottiglia, Filippo; Casu, Laura; L., Bonsignore; Casu, Mariano; Floris, Costantino; Leonti, Marco; J., Gertsch; J., Heilmann | PLANTA MEDICA | - |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile