Università degli Studi di Cagliari
Antimicrobial activity of 10-(diphenylmethylene)-4-azatricyclo[5.2.1.0 2,6]dec-8-ene-3,5-dione derivatives
2010-01-01 Stefanska, J; Bielenica, A; Struga, M; Tyski, S; Kossakowski, J; LA COLLA, P; Tamburini, Elena; Loddo, Roberta
Platinum and palladium-triazole complexes as highly potential antitumor agents
2010-01-01 AL MASOUDI, Na; Abdullah, Bh; Essa, Ah; Loddo, Roberta; AND LA COLLA, P.
1,2-benzisothiazol-3(2h)-one benzenesulfonamides targeting the hiv nucleocapsid proteins are potential microbicide candidates for the prevention of mucosal hiv transmission/acquisition
2010-01-01 Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; Giliberti, Gabriele; Marongiu, E.; Loddo, Roberta; La Colla, P.
Mystery Unveiled: Benzimidazole docks in different domains of HCV and BVDV RdRp
2009-01-01 Shukla, S; Asthana, S; Giliberti, Gabriele; Iuliano, F; Ceccarelli, Matteo; Loddo, Roberta; Ruggerone, P; La Colla, P.
Activity and molecular modeling of a new small molecule active against NNRTI-resistant HIV-1 mutants
2009-01-01 Loddo, Roberta; Pricl, S; Piras, S; Fermeglia, M; LA COLLA, P; Loddo, R.
Biological evaluation of 10-(diphenylmethylene)-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione derivatives
2009-01-01 Stefańska, J; Bielenica, A; Struga, M; Tyski, S; Kossakowski, J; Loddo, Roberta; Ibba, Cristina; Collu, David; Marongiu, E; La Colla, P.
2-Arylbenzimidazoles as Antiviral and Antiproliferative Agents-Part 2
2009-01-01 Vitale, G; Corona, P; Loriga, M; Loddo, Roberta; Paglietti, G; La Colla, P; Busonera, B; Marongiu, E; Collu, David; Loddo, R.
Synthesis and Anti-HIV-1 Activity of 1-Substiuted 6-(3-Cyanobenzoyl) and [(3-Cyanophenyl)fluoromethyl]-5-ethyl-uracils
2009-01-01 Loksha, Ym; Pedersen, Eb; Loddo, Roberta; AND LA COLLA, P.
Anti-HIV evaluation of benzo[d]isothiazole hydrazones
2009-01-01 Vicini, P; Incerti, M; LA COLLA, P; Loddo, Roberta
Hepatitis C: New therapeutic approaches
2009-01-01 Loddo, Roberta; Giliberti, Gabriele; AND PEZZULLO, M.
1,2-benzisothiazol-3(2H)-one benzenesulfonamides as new microbicide candidates for prevention of mucosal HIV infections
2009-01-01 Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; Sanna, Giuseppina; Secci, B; Marongiu, E; Loddo, Roberta; La Colla, P.
Mystery unveiled: benzimidazole docks different domains in Flaviviridae
2009-01-01 Shukla, S; Asthana, S; Giliberti, Gabriele; Iuliano, F; Ceccarelli, Matteo; Loddo, R; Ruggerone, Paolo; La Colla, P.
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Schenone, S; Bruno, O; Borassi, A; LA COLLA, P; Pezzullo, M; Sanna, Giuseppina; Collu, Gabriella; Secci, Barbara; Loddo, Roberta
Antiviral activity of indole derivatives
2009-01-01 Giampieri, M; Balbi, A; Mazzei, M; LA COLLA, P; Ibba, Cristina; Loddo, Roberta
N-acylated and N,N’-diacylated imidazolidine-2-thione derivatives and N,N’-diacylated tetrahydropyrimidine-2(1H)-thione analogues: synthesis and antiproliferative activity
2009-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Rosano, C; LA COLLA, P; Sanna, Giuseppina; Busonera, B; Loddo, Roberta
Synthesis and in vitro antiproliferative activity of new adamantylthiazolyl-1,3,4-oxadiazoles
2009-01-01 Zahid, M; Yasin, Ka; Akhtar, T; Rama, Nh; Hameed, S; AL MASOUDI, Na; Loddo, Roberta; AND LA COLLA, P.
Synthesis of novel uracil non-nucleoside derivatives as potential reverse transcriptase inhibitors of HIV-1
2009-01-01 El Brollosy, Nr; Al Deeb, Oa; El Emam, Aa; Pedersen, Eb; La Colla, P; Collu, G; Sanna, Giuseppina; Loddo, Roberta
Synthesis, pharmacological and antiviral activity of 1,3-thiazepine derivatives
2009-01-01 Struga, M; Kossakowski, J; Koziol, Ae; Kedzierska, E; Fidecka, S; LA COLLA, P; Ibba, Cristina; Collu, G; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Bruno, O; Schenone, S; LA COLLA, P; Collu, Gabriella; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta
Prompt lithiation of 1-dimethylsulfamoylthymine used for the synthesis of 1-allyloxymethyl-6-(a,2,6-trifluorobenzyl)thymine
2009-01-01 Loksha, Ym; Pedersen, Eb; Bond, Ad; LA COLLA, P; Secci, B; Loddo, Roberta
Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters
2009-01-01 Romanowska, J; SZYMANSKA MICHALAK, A; Boryski, J; Stawinski, J; Kraszewski, A; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Secci, Barbara; LA COLLA, P.
Synthesis and evaluation of in vitro biological activity of 4-substituted arylpiperazine derivatives of 1,7,8,9-tetrachloro-10,10-dimethoxy-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
2009-01-01 Kossakowski, J; Pakosinska Parys, M; Struga, M; Dybala, I; E., Koziol A; La Colla, P; Marongiu, Le; Ibba, Cristina; Collu, David; Loddo, Roberta
Synthesis and anti-HIV-1 evaluation of new Sonogashira-modified Emivirine (MKC-442) analogues
2009-01-01 Danel, K; Jørgensen, Pt; Pedersen, Eb; LA COLLA, P; Collu, G; Loddo, Roberta
Antiviral and cytotoxic activities of aminoarylazo compounds and aryltriazene derivatives
2009-01-01 Tonelli, M; Vazzana, I; Tasso, B; Boido, V; Sparatore, F; Fermeglia, M; Paneni, Ms; Posocco, P; Pricl, S; LA COLLA, P; Ibba, Cristina; Secci, Barbara; Collu, G; Loddo, Roberta
Potent flaviviridae inhibitors: targeted finger domain of RdRp
2009-01-01 Asthana, S; Shukla, S; Giliberti, Gabriele; Iuliano, F; Ceccarelli, Matteo; Loddo, Roberta; Ruggerone, Paolo; La Colla, P.
Results on different formulations of an NNRTI candidate (MC 1220) for application as topical microbicide
2009-01-01 Blois, SYLVAIN SERGE DANIEL; Marongiu, E; Sanna, Giuseppina; Collu, G; Secci, B; Giliberti, Gabriele; Loddo, Roberta; Pedersen, E; De Giuli Morghen, C; Stahl Hennig, C; La Colla, P.
Potent flaviviridae inhibitors: targeted finger domain of RdRp.
2009-01-01 Asthana, S; Shukla, S; Giliberti, Gabriele; Iuliano, F; Ceccarelli, Matteo; Loddo, R; Ruggerone, Paolo; La Colla, P.
2-Arylbenzimidazoles as antiviral and antiproliferative agents-Part 1
2008-01-01 Vitale, G; Loddo, Roberta; Loriga, M; Paglietti, G; La Colla, P; Busonera, B; Collu, David; Loddo, R.
Activity of Mannich bases of 7-hydroxycoumarin against Flaviviridae
2008-01-01 Mazzei, M; Nieddu, E; Miele, M; Balbi, A; Ferrone, M; Fermeglia, M; Mazzei, Mt; Pricl, S; La Colla, P; Marongiu, Fabio; Ibba, Cristina; Loddo, Roberta
Design, synthesis and anti Flaviviridae activity of N6-, 5’,3’-O- and 5’,2’-O-substituted adenine nucleoside analogs
2008-01-01 Angusti, A; Manfredini, S; Durini, E; Ciliberti, N; Vertuani, S; Solaroli, N; Pricl, S; Ferrone, M; Fermeglia, M; Loddo, Roberta; Secci, Barbara; Visioli, A; Sanna, T; Collu, Gabriella; Pezzullo, M; LA COLLA, P.
2(3)-aryl-thio(oxy)-methylquinoxaline derivatives: a new class of PGlycoprotein-mediated drug efflux inhibitors
2008-01-01 Loddo, Roberta; Piras, S; Paglietti, G; Pricl, S; LA COLLA, P; Busonera, B; Loddo, R.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Bruno, O; LA COLLA, P; Secci, Barbara; Collu, Gabriella; Loddo, Roberta
In vitro anti-HIV and antitumor activity of new 3,6-disubstituted[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles and Thiadiazine analogues
2008-01-01 AL SOUD, Ya; AL MASOUDI, Na; Loddo, Roberta; LA COLLA, P.
Synthesis and in vitro antiproliferative activity of new benzothiazole derivatives
2008-01-01 AL SOUD, Ya; AL SADONI, Hh; Saeed, B; Jaber, Ih; BENI KHALID, Mo; AL MASOUDI, Na; ABDUL KADIR, T; LA COLLA, P; Busonera, B; Sanna, T; Loddo, Roberta
Synthesis and anti-HIV-1 evaluation of 1,5-disubstituted pyrimidine-2,4-diones
2008-01-01 Loksha, Ym; Globisch, D; Pedersen, Eb; LA COLLA, P; Collu, Gabriella; Loddo, Roberta
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Bruno, O; LA COLLA, P; Casula, L; Collu, Gabriella; Sanna, Giuseppina; Loddo, Roberta
Antiviral activity of benzimidazole derivatives. I. Antiviral activity of 1-substituted-2-[(benzotriazol-1/2-yl)methyl]benzimidazoles
2008-01-01 Tonelli, M; Paglietti, G; Boido, V; Sparatore, F; Marongiu, Fabio; Marongiu, E; La Colla, P; Loddo, Roberta
In vitro antitumor and antiviral activities of new benzothiazole and 1,3,4-oxadiazole-2-thione derivatives
2008-01-01 Akhtar, T; Hameed, S; AL MASOUDI, Na; Loddo, Roberta; LA COLLA, P.
Antimicrobial and cytotoxic arylazoenamines. Part III: antiviral activity of selected classes of arylazoenamines
2008-01-01 Tonelli, M; Boido, V; Canu, C; Sparatore, A; Sparatore, F; Paneni, Ms; Fermeglia, M; Pricl, S; La Colla, P; Casula, L; Ibba, Cristina; Collu, David; Loddo, Roberta
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Fossa, P; LA COLLA, P; Sanna, Giuseppina; Collu, G; Loddo, Roberta
Synthesis and antiviral activity of new dimeric inhibitors against HIV-1
2008-01-01 Danel, K; Larsen, Lm; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta
Synthesis and antiviral evaluation of 6-(trifluoromethylbenzyl) and 6-(fluorobenzyl) analogues of HIV drugs Emivirine and GCA-186
2008-01-01 EL BROLLOSY, Nr; Sørensen, Er; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta
In vitro evaluation of the anti-HIV-1 activity of Liposomes and gel ingredients
2008-01-01 Loddo, Roberta; Sanna, Giuseppina; Collu, G; Busonera, B; Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; La Colla, P.
Benzimidazoles as potent non nucleosidic inhibitors of Respiratory Syncytial Virus
2008-01-01 Iuliano, F; Collu, D; Giliberti, Gabriele; Ibba, C; Casula, L; Loddo, Roberta; La Colla, P.
Novel Synthesis and Anti-HIV-1 Activity of 2-Arylthio-6-benzyl-2,3-dihydro-1H-pyrimidin-4-ones (Aryl S-DABOs)
2007-01-01 Aly, Yl; Pedersen, Eb; LA COLLA, P; Loddo, Roberta
Synthesis and in vitro antiviral studies of bis(pivaloyloxymethyl)ester derivative of 9-[((phosphonomethyl)aziridin-1-yl)methyl]adenine(PMAMA) and analogues
2007-01-01 ABU SHEIKHA, Gm; Bkhaitan, Mm; AL HOURANI, Ra; Qaisi, Am; Loddo, Roberta; LA COLLA, P.
Design, synthesis, and preliminary in vitro and in silico antiviral activity of [4,7]phenantrolines and 1-oxo-1,4-dihydro- [4,7]phenantrolines against single-stranded positive-sense RNA genome viruses
2007-01-01 Loddo, Roberta; Loriga, M; Paglietti, G; Ferrone, M; Fermeglia, M; Pricl, S; Sanna, T; Ibba, Cristina; LA COLLA, P; Loddo, R.
Synthesis and anti-HIV-1 activity of new MKC-442 analogues with an alkynyl-substituted 6-benzyl group
2007-01-01 Aly, Yl; Pedersen, Eb; LA COLLA, P; Loddo, Roberta
Synthesis and anti-Picornaviridae in vitro activity of a new class of helicase inhibitors the N,N’-bis[4-(1H(2H)-benzotriazol-1(2)-yl)phenyl]alkyldicarboxamides
2007-01-01 Loddo, Roberta; Loriga, M; Piras, S; Paglietti, G; Ferrone, M; Fermeglia, M; Pricl, S; LA COLLA, P; Collu, Gabriella; Sanna, T.; Loddo, R.
Synthesis of some novel 2,6-disubstituted pyridazin-3-ones as TMC120 analogues
2007-01-01 Loksha, Ym; Pedersen, Eb; LA COLLA, P; Loddo, Roberta
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