Maria Paola Castelli
Correlations between Gustatory, Olfactory, Cognitive Function, and Age in Healthy Women
2024-01-01 Sanna, Fabrizio; Castelli, MARIA PAOLA; Mostallino, Rafaela; Loy, Francesco; Masala, Carla
Regioselective synthesis of new EWG-Bearing 3-benzoyl-2-phenylbenzofurans by one-pot intramolecular acylation/thermal cyclization of phosphoranes and their CB1 antagonist activity
2024-01-01 Begala, Michela; Mancinelli, Michele; Mostallino, Rafaela; Castelli, MARIA PAOLA; Delogu, GIOVANNA LUCIA
Implications of disease-modifying therapies for multiple sclerosis on immune cells and response to COVID-19 vaccination
2024-01-01 Orrù, Valeria; Serra, Valentina; Marongiu, Michele; Lai, Sandra; Lodde, Valeria; Zoledziewska, Magdalena; Steri, Maristella; Loizedda, Annalisa; Lobina, Monia; Piras, Maria Grazia; Virdis, Francesca; Delogu, Giuseppe; Marini, Maria Giuseppina; Mingoia, Maura; Floris, Matteo; Masala, Marco; Castelli, M Paola; Mostallino, Rafaela; Frau, Jessica; Lorefice, Lorena; Farina, Gabriele; Fronza, Marzia; Carmagnini, Daniele; Carta, Elisa; Pilotto, Silvy; Chessa, Paola; Devoto, Marcella; Castiglia, Paolo; Solla, Paolo; Zarbo, Roberto Ignazio; Idda, Maria Laura; Pitzalis, Maristella; Cocco, Eleonora; Fiorillo, Edoardo; Cucca, Francesco
Immune and glial cell alterations in the rat brain after repeated exposure to the synthetic cannabinoid JWH-018
2024-01-01 Pintori, Nicholas; Mostallino, Rafaela; Spano, Enrica; Orrù, Valeria; Piras, Maria Grazia; Castelli, Maria Paola; De Luca, Maria Antonietta
Adolescent self-administration of the synthetic cannabinoid receptor agonist JWH-018 induces neurobiological and behavioral alterations in adult male mice
2023-01-01 Margiani, Giulia; Castelli, Maria Paola; Pintori, Nicholas; Frau, Roberto; Ennas, Maria Grazia; Pagano Zottola, Antonio C.; Orrù, Valeria; Serra, Valentina; Fiorillo, Edoardo; Fadda, Paola; Marsicano, Giovanni; De Luca, Maria Antonietta
Maternal immune activation impairs endocannabinoid signaling in the mesolimbic system of adolescent male offspring
2023-01-01 Santoni, Michele; Sagheddu, Claudia; Serra, Valeria; Mostallino, Rafaela; Paola Castelli, Maria; Pisano, Francesco; Scherma, Maria; Fadda, Paola; Muntoni, Anna Lisa; Zamberletti, Erica; Rubino, Tiziana; Melis, Miriam; Pistis, Marco
Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists
2022-01-01 De Luca, Maria Antonietta; Tocco, Graziella; Mostallino, Rafaela; Laus, Antonio; Caria, Francesca; Musa, Aurora; Pintori, Nicholas; Ucha, Marcos; Poza, Celia; Ambrosio, Emilio; Di Chiara, Gaetano; Castelli, M Paola
Adolescent self-administration of the synthetic cannabinoid receptor agonist JWH-018 induces neurobiological and behavioral alterations in adult male mice
2022-01-01 Margiani, Giulia; Castelli, Maria Paola; Pintori, Nicholas; Frau, Roberto; Ennas, Maria Grazia; Orrù, Valeria; Serra, Valentina; Fiorillo, Edoardo; Fadda, Paola; Marsicano, Giovanni; De Luca, Maria Antonietta
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists
2022-01-01 Tocco, Graziella; Laus, Antonio; Vanejevs, Maksims; Ture, Anastasija; Mostallino, Rafaela; Pintori, Nicholas; De Luca, Maria Antonietta; Castelli, M. Paola; Di Chiara, Gaetano
Human neuronal cell lines as an in vitro toxicological tool for the evaluation of novel psychoactive substances
2021-01-01 Sogos, V.; Caria, P.; Porcedda, C.; Mostallino, R.; Piras, F.; Miliano, C.; De Luca, M. A.; Castelli, M. P.
Repeated exposure to JWH-018 induces adaptive changes in the mesolimbic and mesocortical dopamine pathways, glial cells alteration and behavioural correlates
2021-01-01 Pintori, Nicholas; Castelli, Maria Paola; Miliano, Cristina; Simola, Nicola; Fadda, Paola; Fattore, Liana; Scherma, Maria; Ennas, Maria Grazia; Mostallino, Rafaela; Flore, Giovanna; De Felice, Marta; Sagheddu, Claudia; Pistis, Marco; Di Chiara, Gaetano; De Luca, Maria Antonietta
COR758, a negative allosteric modulator of GABAB receptors
2021-01-01 Porcu, A.; Mostallino, R.; Serra, V.; Melis, M.; Sogos, V.; Beggiato, S.; Ferraro, L.; Manetti, F.; Gianibbi, B.; Bettler, B.; Corelli, F.; Mugnaini, C.; Castelli, M. P.
Structure optimization of positive allosteric modulators of GABAB receptors led to the unexpected discovery of antagonists/potential negative allosteric modulators
2020-01-01 Mugnaini, C.; Brizzi, A.; Mostallino, R.; Castelli, M. P.; Corelli, F.
Sex and gender differences in the effects of novel psychoactive substances
2020-01-01 Fattore, Liana; Marti, Matteo; Mostallino, Rafaela; Castelli, Maria Paola
The GABAB receptor positive allosteric modulator COR659: in vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives
2020-01-01 Ferlenghi, Francesca; Maccioni, Paola; Mugnaini, Claudia; Brizzi, Antonella; Fara, Federica; Mostallino, Rafaela; Castelli, Maria Paola; Colombo, Giancarlo; Mor, Marco; Vacondio, Federica; Corelli, Federico
Impaired brain endocannabinoid tone in the activity-based model of anorexia nervosa
2019-01-01 Collu, R.; Scherma, M.; Piscitelli, F.; Giunti, E.; Satta, V.; Castelli, M. P.; Verde, R.; Fratta, W.; Bisogno, T.; Fadda, P.
Neurochemical and Behavioral Profiling in Male and Female Rats of the Psychedelic Agent 25I-NBOMe
2019-01-01 Miliano, Cristina; Marti, Matteo; Pintori, Nicholas; Castelli, Maria Paola; Tirri, Micaela; Arfè, Raffaella; De Luca, Maria Antonietta
Predisposition to alcohol drinking and alcohol consumption alter expression of calcitonin gene-related peptide, neuropeptide Y, and microglia in bed nucleus of stria terminalis in a subnucleus-specific manner
2019-01-01 Rossetti, Ilaria; Zambusi, Laura; Maccioni, Paola; Sau, Roberta; Provini, Luciano; Castelli, MARIA PAOLA; Gonciarz, Krzysztof; Colombo, Giancarlo; Morara, Stefano
Limited access to a high fat diet alters endocannabinoid tone in female rats
2018-01-01 Satta, Valentina; Scherma, Maria; Piscitelli, Fabiana; Usai, Paolo; Castelli, M Paola; Bisogno, Tiziana; Fratta, Walter; Fadda, Paola
In vitro functional characterization of GET73 as possible negative allosteric modulator of metabotropic glutamate receptor 5
2018-01-01 Beggiato, Sarah; Borelli, Andrea C.; Tomasini, Maria C.; Castelli, MARIA PAOLA; Pintori, Nicholas; Cacciaglia, Roberto; Loche, Antonella; Ferraro, LUCA NICOLA
Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a G alpha(i/o) protein inhibitor
2018-01-01 Porcu, Alessandra; Melis, Miriam; Turecek, Rostislav; Ullrich, Celine; Mocci, Ignazia; Bettler, Bernhard; Luigi Gessa, Gian; Castelli, MARIA PAOLA
Suppressing effect of saikosaponin A, an active ingredient of Bupleurum falcatum, on chocolate self-administration and reinstatement of chocolate seeking in rats
2017-01-01 Lorrai, Irene; Maccioni, Paola; Carai, MAURO ANTONIO MARIA; Capra, Alessandro; Castelli, MARIA PAOLA; Riva, Antonella; Morazzoni, Paolo; Gessa, Gian Luigi; Colombo, Giancarlo
Cannabis and the Use of Amphetamine-Like Substances
2017-01-01 Porcu, Alessandra; Castelli, MARIA PAOLA
Native CB1 receptor affinity, intrinsic activity and accumbens shell dopamine stimulant properties of third generation SPICE/K2 cannabinoids: BB-22, 5F-PB-22, 5F-AKB-48 and STS-135
2016-01-01 DE LUCA, MARIA ANTONIETTA; Castelli, MARIA PAOLA; Loi, B; Porcu, Alessandra; Martorelli, Mariella; Miliano, Cristina; Kellett, K; Davidson, C; Stair, Jl; Schifano, F; DI CHIARA, Gaetano
Influence of caffeine on 3,4-methylenedioxymethamphetamine-induced dopaminergic neuron degeneration and neuroinflammation is age-dependent
2016-01-01 Frau, Lucia; Costa, Giulia; Porceddu, Pier Francesca; Khairnar, Amit; Castelli, Maria Paola; Ennas, Maria Grazia; Madeddu, Camilla; Wardas, Jadwiga; Morelli, Micaela
In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator
2016-01-01 Porcu, Alessandra; Lobina, Carla; Giunta, Daniela; Solinas, Maurizio; Mugnaini, Claudia; Castelli, MARIA PAOLA
α2A adrenergic receptors highly expressed in mesoprefrontal dopamine neurons
2016-01-01 Castelli, MARIA PAOLA; Spiga, Saturnino; Perra, Andrea; Madeddu, Camilla; Mulas, Giovanna; Ennas, MARIA GRAZIA; Gessa, Gl
Distribution and localization of the GABAB receptor
2016-01-01 Castelli, MARIA PAOLA; Gessa, Gian Luigi
The Role of the Endocannabinoid System in Eating Disorders: Neurochemical and Behavioural Preclinical Evidence.
2014-01-01 Scherma, Maria; Fattore, L; Castelli, MARIA PAOLA; Fratta, Walter; Fadda, Paola
The agression and behavioral abnormalities associated with monoamine oxidase A deficiency are rescued by acute inhibition of serotonin reuptake.
2014-01-01 Godar, Sc; Bortolato, M; Castelli, MARIA PAOLA; Casti, Alberto; Casu, A; Chen, K; Ennas, MARIA GRAZIA; Tambaro, S; Shih, Jc
Synthesis, structural properties, and pharmacological evaluation of 2-(acylamino)-thiophene-3-carboxamides and analogues thereof
2014-01-01 Mugnaini, C; Pedani, V; Giunta, D; Secchi, B; Solinas, M; Casti, Alberto; Castelli, MARIA PAOLA; Giorgi, G; Corelli, F.
Enhanced endocannabinoid-mediated modulation of rostromedial tegmental nucleus drive onto dopamine neurons in sardinian alcohol-preferring rats
2014-01-01 Melis, Miriam; Sagheddu, Claudia; De Felice, M; Casti, Alberto; Madeddu, Camilla; Spiga, Saturnino; Muntoni, Al; Mackie, K; Marsicano, G; Colombo, G; Castelli, MARIA PAOLA; Pistis, Marco
Male and Female Rats Differ in Brain Cannabinoid CB1 Receptor Density and Function and in Behavioural Traits Predisposing To Drug Addiction: Effect of Ovarian Hormones.
2014-01-01 Castelli, MARIA PAOLA; Fadda, Paola; Casu, A; Spano, Ms; Casti, Alberto; Fratta, Walter; Fattore, L.
Δ9-Tetrahydrocannabinol prevents methamphetamine-induced neurotoxicity
2014-01-01 Castelli, MARIA PAOLA; Madeddu, Camilla; Casti, Alberto; Casu, A; Casti, P; Scherma, Maria; Fattore, L; Fadda, Paola; Ennas, MARIA GRAZIA
Regional distribution of 5α-reductase type 2 in the adult rat brain: An immunohistochemical analysis
2013-01-01 Castelli, MARIA PAOLA; Casti, Alberto; Casu, A; Frau, Roberto; Bortolato, M; Spiga, Saturnino; Ennas, MARIA GRAZIA
Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor
2013-01-01 Mugnaini, C; Pedani, V; Casu, A; Lobina, C; Casti, Alberto; Maccioni, P; Porcu, Alessandra; Giunta, D; Lamponi, S; Solinas, M; Dragoni, S; Valoti, M; Colombo, G; Castelli, MARIA PAOLA; Gessa, Gl; Corelli, F.
The new compound GET73, N-[(4-trifluoromethyl)benzyl]4-methoxybutyramide, regulates hippocampal aminoacidergic transmission possibly via an allosteric modulation of mGlu5 receptor. Behavioural evidence of its "anti-alcohol" and anxiolytic properties.
2013-01-01 Ferraro, L.; Loche, A.; Beggiato, S.; Tomasini, M. C.; Antonelli, T.; Colombo, G.; Lobina, C.; Carai, M. A. M.; Porcu, Alessandra; Castelli, MARIA PAOLA; Clerici, F.; Borelli, A. C.; Cacciaglia, R.; Tanganelli, S.
PPARα regulates cholinergic-driven activity of midbrain dopamine neurons via a novel mechanism involving α7 nicotinic acetylcholine receptors.
2013-01-01 Melis, Miriam; Scheggi, S; Carta, Gianfranca; Madeddu, Camilla; Lecca, Salvatore; Luchicchi, A; Cadeddu, Francesca; Frau, Roberto; Fattore, L; Fadda, Paola; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA; Fratta, Walter; Schilstrom, B; Banni, Sebastiano; De Montis, Mg; Pistis, Marco
NMDA receptors mediate the role of monoamine oxidase A in pathological aggression
2012-01-01 Godar, Sc; Bortolato, M; Melis, M; Soggiu, A; Roncada, P; Casu, A; Flore, G; Chen, K; Frau, Roberto; Urbani, A; Castelli, MARIA PAOLA; Devoto, Paola; Shih, Jc
Inhibition of steroid 5-alpha reductase reduces marble-burying responses in mice
2012-01-01 Bini, V; Frau, Roberto; Paba, S; Collu, Maria; Castelli, MARIA PAOLA; Devoto, Paola; Bortolato, M.
Reversible disruption of pre-pulse inhibition in hypomorphic-inducible and reversible CB1-/- mice
2012-01-01 Marongiu, Mfranca; Poddie, D; Porcu, S; Manchinu, Mf; Castelli, MARIA PAOLA; Sogos, Valeria; Bini, V; Frau, Roberto; Caredda, E; Collu, Maria; Ristaldi, Ms
Anti-Alcohol and Anxiolytic Properties of a New Chemical Entity, GET73.
2012-01-01 Loche, A; Simonetti, F; Lobina, C; Carai, Ma; Colombo, G; Castelli, MARIA PAOLA; Barone, D; Cacciaglia, R.
Characterization of COR627 and COR628, Two Novel Positive Allosteric Modulators of the GABAB Receptor.
2012-01-01 Castelli, MARIA PAOLA; Casu, A; Casti, P; Lobina, C; Carai, Ma; Colombo, G; Solinas, M; Giunta, D; Mugnaini, C; Pasquini, S; Tafi, A; Brogi, S; Gessa, Gl; Corelli, F.
NMDARs mediate the role of monoamine oxidase A in pathological aggression
2012-01-01 Bortolato, M; Godar, Sc; Melis, Miriam; Soggiu, A; Roncada, P; Casu, A; Flore, G; Chen, K; Frau, Roberto; Urbani, A; Castelli, MARIA PAOLA; Devoto, Paola; Shih, Jc
Localization of steroid 5α-reductase type 2 isozyme in the adult rat brain
2011-01-01 Casti, A; Casu, A; Casti, P; Frau, Roberto; Bortolato, M; Spiga, Saturnino; Castelli, MARIA PAOLA; Ennas, Mg
Effects of drugs of abuse on putative rostromedial tegmental neurons, inhibitory afferents to midbrain dopamine cells
2011-01-01 Lecca, Salvatore; Melis, Miriam; Luchicchi, A; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA; Muntoni A., L; Pistis, Marco
Adolescent exposure to nicotine and/or the cannabinoid agonist CP 55,940 induces gender-dependent long lasting memory impairments and changes in brain nicotinic and CB1 cannabinoid receptors
2011-01-01 Mateos, B; Borcel, E; Loriga, R; Luesu, W; Bini, V; Llorente, R; Castelli, MARIA PAOLA; Viveros, Mp
Methamphetamine neurotoxicity increases brain expression and alters behavioral functions of CB(1) cannabinoid receptors
2010-01-01 Bortolato, M; Frau, Roberto; Bini, V; Luesu, W; Loriga, Roberta; Collu, Maria; Gessa, Gl; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA
Changes induced by acute toxic dose (ATD) of methanphetamine (METH) on cannabinoid CB1 receptors: An immunocytochemistry study
2009-01-01 Luesu, W; Bini, V; Tuveri, B; Loriga, R; Castelli, MARIA PAOLA; Ennas, MARIA GRAZIA
Persistent increase in CB1 receptor and amnestic effect of cannabinoid by methamphetamine
2009-01-01 Frau, Roberto; V., Bini; W., Luesu; Loriga, Roberta; Collu, Maria; G. L., Gessa; M. G., Ennas; M., Bortolato; Castelli, MARIA PAOLA
Title | Issue Date | Author(s) | Journal | Publisher |
---|---|---|---|---|
Correlations between Gustatory, Olfactory, Cognitive Function, and Age in Healthy Women | 1-Jan-2024 | Sanna, Fabrizio; Castelli, MARIA PAOLA; Mostallino, Rafaela; Loy, Francesco; Masala, Carla | NUTRIENTS | - |
Regioselective synthesis of new EWG-Bearing 3-benzoyl-2-phenylbenzofurans by one-pot intramolecular acylation/thermal cyclization of phosphoranes and their CB1 antagonist activity | 1-Jan-2024 | Begala, Michela; Mancinelli, Michele; Mostallino, Rafaela; Castelli, MARIA PAOLA; Delogu, GIOVANNA LUCIA | TETRAHEDRON | - |
Implications of disease-modifying therapies for multiple sclerosis on immune cells and response to COVID-19 vaccination | 1-Jan-2024 | Orrù, Valeria; Serra, Valentina; Marongiu, Michele; Lai, Sandra; Lodde, Valeria; Zoledziewska, Magdalena; Steri, Maristella; Loizedda, Annalisa; Lobina, Monia; Piras, Maria Grazia; Virdis, Francesca; Delogu, Giuseppe; Marini, Maria Giuseppina; Mingoia, Maura; Floris, Matteo; Masala, Marco; Castelli, M Paola; Mostallino, Rafaela; Frau, Jessica; Lorefice, Lorena; Farina, Gabriele; Fronza, Marzia; Carmagnini, Daniele; Carta, Elisa; Pilotto, Silvy; Chessa, Paola; Devoto, Marcella; Castiglia, Paolo; Solla, Paolo; Zarbo, Roberto Ignazio; Idda, Maria Laura; Pitzalis, Maristella; Cocco, Eleonora; Fiorillo, Edoardo; Cucca, Francesco | FRONTIERS IN IMMUNOLOGY | - |
Immune and glial cell alterations in the rat brain after repeated exposure to the synthetic cannabinoid JWH-018 | 1-Jan-2024 | Pintori, Nicholas; Mostallino, Rafaela; Spano, Enrica; Orrù, Valeria; Piras, Maria Grazia; Castelli, Maria Paola; De Luca, Maria Antonietta | JOURNAL OF NEUROIMMUNOLOGY | - |
Adolescent self-administration of the synthetic cannabinoid receptor agonist JWH-018 induces neurobiological and behavioral alterations in adult male mice | 1-Jan-2023 | Margiani, Giulia; Castelli, Maria Paola; Pintori, Nicholas; Frau, Roberto; Ennas, Maria Grazia; Pagano Zottola, Antonio C.; Orrù, Valeria; Serra, Valentina; Fiorillo, Edoardo; Fadda, Paola; Marsicano, Giovanni; De Luca, Maria Antonietta | PSYCHOPHARMACOLOGY | - |
Maternal immune activation impairs endocannabinoid signaling in the mesolimbic system of adolescent male offspring | 1-Jan-2023 | Santoni, Michele; Sagheddu, Claudia; Serra, Valeria; Mostallino, Rafaela; Paola Castelli, Maria; Pisano, Francesco; Scherma, Maria; Fadda, Paola; Muntoni, Anna Lisa; Zamberletti, Erica; Rubino, Tiziana; Melis, Miriam; Pistis, Marco | BRAIN BEHAVIOR AND IMMUNITY | - |
Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists | 1-Jan-2022 | De Luca, Maria Antonietta; Tocco, Graziella; Mostallino, Rafaela; Laus, Antonio; Caria, Francesca; Musa, Aurora; Pintori, Nicholas; Ucha, Marcos; Poza, Celia; Ambrosio, Emilio; Di Chiara, Gaetano; Castelli, M Paola | NEUROPHARMACOLOGY | - |
Adolescent self-administration of the synthetic cannabinoid receptor agonist JWH-018 induces neurobiological and behavioral alterations in adult male mice | 1-Jan-2022 | Margiani, Giulia; Castelli, Maria Paola; Pintori, Nicholas; Frau, Roberto; Ennas, Maria Grazia; Orrù, Valeria; Serra, Valentina; Fiorillo, Edoardo; Fadda, Paola; Marsicano, Giovanni; De Luca, Maria Antonietta | PSYCHOPHARMACOLOGY | - |
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists | 1-Jan-2022 | Tocco, Graziella; Laus, Antonio; Vanejevs, Maksims; Ture, Anastasija; Mostallino, Rafaela; Pintori, Nicholas; De Luca, Maria Antonietta; Castelli, M. Paola; Di Chiara, Gaetano | ARCHIV DER PHARMAZIE | - |
Human neuronal cell lines as an in vitro toxicological tool for the evaluation of novel psychoactive substances | 1-Jan-2021 | Sogos, V.; Caria, P.; Porcedda, C.; Mostallino, R.; Piras, F.; Miliano, C.; De Luca, M. A.; Castelli, M. P. | INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES | - |
Repeated exposure to JWH-018 induces adaptive changes in the mesolimbic and mesocortical dopamine pathways, glial cells alteration and behavioural correlates | 1-Jan-2021 | Pintori, Nicholas; Castelli, Maria Paola; Miliano, Cristina; Simola, Nicola; Fadda, Paola; Fattore, Liana; Scherma, Maria; Ennas, Maria Grazia; Mostallino, Rafaela; Flore, Giovanna; De Felice, Marta; Sagheddu, Claudia; Pistis, Marco; Di Chiara, Gaetano; De Luca, Maria Antonietta | BRITISH JOURNAL OF PHARMACOLOGY | - |
COR758, a negative allosteric modulator of GABAB receptors | 1-Jan-2021 | Porcu, A.; Mostallino, R.; Serra, V.; Melis, M.; Sogos, V.; Beggiato, S.; Ferraro, L.; Manetti, F.; Gianibbi, B.; Bettler, B.; Corelli, F.; Mugnaini, C.; Castelli, M. P. | NEUROPHARMACOLOGY | - |
Structure optimization of positive allosteric modulators of GABAB receptors led to the unexpected discovery of antagonists/potential negative allosteric modulators | 1-Jan-2020 | Mugnaini, C.; Brizzi, A.; Mostallino, R.; Castelli, M. P.; Corelli, F. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Sex and gender differences in the effects of novel psychoactive substances | 1-Jan-2020 | Fattore, Liana; Marti, Matteo; Mostallino, Rafaela; Castelli, Maria Paola | BRAIN SCIENCES | - |
The GABAB receptor positive allosteric modulator COR659: in vitro metabolism, in vivo pharmacokinetics in rats, synthesis and pharmacological characterization of metabolically protected derivatives | 1-Jan-2020 | Ferlenghi, Francesca; Maccioni, Paola; Mugnaini, Claudia; Brizzi, Antonella; Fara, Federica; Mostallino, Rafaela; Castelli, Maria Paola; Colombo, Giancarlo; Mor, Marco; Vacondio, Federica; Corelli, Federico | EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES | - |
Impaired brain endocannabinoid tone in the activity-based model of anorexia nervosa | 1-Jan-2019 | Collu, R.; Scherma, M.; Piscitelli, F.; Giunti, E.; Satta, V.; Castelli, M. P.; Verde, R.; Fratta, W.; Bisogno, T.; Fadda, P. | INTERNATIONAL JOURNAL OF EATING DISORDERS | - |
Neurochemical and Behavioral Profiling in Male and Female Rats of the Psychedelic Agent 25I-NBOMe | 1-Jan-2019 | Miliano, Cristina; Marti, Matteo; Pintori, Nicholas; Castelli, Maria Paola; Tirri, Micaela; Arfè, Raffaella; De Luca, Maria Antonietta | FRONTIERS IN PHARMACOLOGY | - |
Predisposition to alcohol drinking and alcohol consumption alter expression of calcitonin gene-related peptide, neuropeptide Y, and microglia in bed nucleus of stria terminalis in a subnucleus-specific manner | 1-Jan-2019 | Rossetti, Ilaria; Zambusi, Laura; Maccioni, Paola; Sau, Roberta; Provini, Luciano; Castelli, MARIA PAOLA; Gonciarz, Krzysztof; Colombo, Giancarlo; Morara, Stefano | FRONTIERS IN CELLULAR NEUROSCIENCE | - |
Limited access to a high fat diet alters endocannabinoid tone in female rats | 1-Jan-2018 | Satta, Valentina; Scherma, Maria; Piscitelli, Fabiana; Usai, Paolo; Castelli, M Paola; Bisogno, Tiziana; Fratta, Walter; Fadda, Paola | FRONTIERS IN NEUROSCIENCE | - |
In vitro functional characterization of GET73 as possible negative allosteric modulator of metabotropic glutamate receptor 5 | 1-Jan-2018 | Beggiato, Sarah; Borelli, Andrea C.; Tomasini, Maria C.; Castelli, MARIA PAOLA; Pintori, Nicholas; Cacciaglia, Roberto; Loche, Antonella; Ferraro, LUCA NICOLA | FRONTIERS IN PHARMACOLOGY | - |
Rimonabant, a potent CB1 cannabinoid receptor antagonist, is a G alpha(i/o) protein inhibitor | 1-Jan-2018 | Porcu, Alessandra; Melis, Miriam; Turecek, Rostislav; Ullrich, Celine; Mocci, Ignazia; Bettler, Bernhard; Luigi Gessa, Gian; Castelli, MARIA PAOLA | NEUROPHARMACOLOGY | - |
Suppressing effect of saikosaponin A, an active ingredient of Bupleurum falcatum, on chocolate self-administration and reinstatement of chocolate seeking in rats | 1-Jan-2017 | Lorrai, Irene; Maccioni, Paola; Carai, MAURO ANTONIO MARIA; Capra, Alessandro; Castelli, MARIA PAOLA; Riva, Antonella; Morazzoni, Paolo; Gessa, Gian Luigi; Colombo, Giancarlo | NEUROSCIENCE LETTERS | - |
Cannabis and the Use of Amphetamine-Like Substances | 1-Jan-2017 | Porcu, Alessandra; Castelli, MARIA PAOLA | - | Elsevier |
Native CB1 receptor affinity, intrinsic activity and accumbens shell dopamine stimulant properties of third generation SPICE/K2 cannabinoids: BB-22, 5F-PB-22, 5F-AKB-48 and STS-135 | 1-Jan-2016 | DE LUCA, MARIA ANTONIETTA; Castelli, MARIA PAOLA; Loi, B; Porcu, Alessandra; Martorelli, Mariella; Miliano, Cristina; Kellett, K; Davidson, C; Stair, Jl; Schifano, F; DI CHIARA, Gaetano | NEUROPHARMACOLOGY | - |
Influence of caffeine on 3,4-methylenedioxymethamphetamine-induced dopaminergic neuron degeneration and neuroinflammation is age-dependent | 1-Jan-2016 | Frau, Lucia; Costa, Giulia; Porceddu, Pier Francesca; Khairnar, Amit; Castelli, Maria Paola; Ennas, Maria Grazia; Madeddu, Camilla; Wardas, Jadwiga; Morelli, Micaela | JOURNAL OF NEUROCHEMISTRY | - |
In vitro and in vivo pharmacological characterization of SSD114, a novel GABAB positive allosteric modulator | 1-Jan-2016 | Porcu, Alessandra; Lobina, Carla; Giunta, Daniela; Solinas, Maurizio; Mugnaini, Claudia; Castelli, MARIA PAOLA | EUROPEAN JOURNAL OF PHARMACOLOGY | - |
α2A adrenergic receptors highly expressed in mesoprefrontal dopamine neurons | 1-Jan-2016 | Castelli, MARIA PAOLA; Spiga, Saturnino; Perra, Andrea; Madeddu, Camilla; Mulas, Giovanna; Ennas, MARIA GRAZIA; Gessa, Gl | NEUROSCIENCE | - |
Distribution and localization of the GABAB receptor | 1-Jan-2016 | Castelli, MARIA PAOLA; Gessa, Gian Luigi | - | Springer |
The Role of the Endocannabinoid System in Eating Disorders: Neurochemical and Behavioural Preclinical Evidence. | 1-Jan-2014 | Scherma, Maria; Fattore, L; Castelli, MARIA PAOLA; Fratta, Walter; Fadda, Paola | CURRENT PHARMACEUTICAL DESIGN | - |
The agression and behavioral abnormalities associated with monoamine oxidase A deficiency are rescued by acute inhibition of serotonin reuptake. | 1-Jan-2014 | Godar, Sc; Bortolato, M; Castelli, MARIA PAOLA; Casti, Alberto; Casu, A; Chen, K; Ennas, MARIA GRAZIA; Tambaro, S; Shih, Jc | JOURNAL OF PSYCHIATRIC RESEARCH | - |
Synthesis, structural properties, and pharmacological evaluation of 2-(acylamino)-thiophene-3-carboxamides and analogues thereof | 1-Jan-2014 | Mugnaini, C; Pedani, V; Giunta, D; Secchi, B; Solinas, M; Casti, Alberto; Castelli, MARIA PAOLA; Giorgi, G; Corelli, F. | RSC ADVANCES | - |
Enhanced endocannabinoid-mediated modulation of rostromedial tegmental nucleus drive onto dopamine neurons in sardinian alcohol-preferring rats | 1-Jan-2014 | Melis, Miriam; Sagheddu, Claudia; De Felice, M; Casti, Alberto; Madeddu, Camilla; Spiga, Saturnino; Muntoni, Al; Mackie, K; Marsicano, G; Colombo, G; Castelli, MARIA PAOLA; Pistis, Marco | THE JOURNAL OF NEUROSCIENCE | - |
Male and Female Rats Differ in Brain Cannabinoid CB1 Receptor Density and Function and in Behavioural Traits Predisposing To Drug Addiction: Effect of Ovarian Hormones. | 1-Jan-2014 | Castelli, MARIA PAOLA; Fadda, Paola; Casu, A; Spano, Ms; Casti, Alberto; Fratta, Walter; Fattore, L. | CURRENT PHARMACEUTICAL DESIGN | - |
Δ9-Tetrahydrocannabinol prevents methamphetamine-induced neurotoxicity | 1-Jan-2014 | Castelli, MARIA PAOLA; Madeddu, Camilla; Casti, Alberto; Casu, A; Casti, P; Scherma, Maria; Fattore, L; Fadda, Paola; Ennas, MARIA GRAZIA | PLOS ONE | - |
Regional distribution of 5α-reductase type 2 in the adult rat brain: An immunohistochemical analysis | 1-Jan-2013 | Castelli, MARIA PAOLA; Casti, Alberto; Casu, A; Frau, Roberto; Bortolato, M; Spiga, Saturnino; Ennas, MARIA GRAZIA | PSYCHONEUROENDOCRINOLOGY | - |
Synthesis and pharmacological characterization of 2-(acylamino)thiophene derivatives as metabolically stable, orally effective, positive allosteric modulators of the GABAB receptor | 1-Jan-2013 | Mugnaini, C; Pedani, V; Casu, A; Lobina, C; Casti, Alberto; Maccioni, P; Porcu, Alessandra; Giunta, D; Lamponi, S; Solinas, M; Dragoni, S; Valoti, M; Colombo, G; Castelli, MARIA PAOLA; Gessa, Gl; Corelli, F. | JOURNAL OF MEDICINAL CHEMISTRY | - |
The new compound GET73, N-[(4-trifluoromethyl)benzyl]4-methoxybutyramide, regulates hippocampal aminoacidergic transmission possibly via an allosteric modulation of mGlu5 receptor. Behavioural evidence of its "anti-alcohol" and anxiolytic properties. | 1-Jan-2013 | Ferraro, L.; Loche, A.; Beggiato, S.; Tomasini, M. C.; Antonelli, T.; Colombo, G.; Lobina, C.; Carai, M. A. M.; Porcu, Alessandra; Castelli, MARIA PAOLA; Clerici, F.; Borelli, A. C.; Cacciaglia, R.; Tanganelli, S. | CURRENT MEDICINAL CHEMISTRY | - |
PPARα regulates cholinergic-driven activity of midbrain dopamine neurons via a novel mechanism involving α7 nicotinic acetylcholine receptors. | 1-Jan-2013 | Melis, Miriam; Scheggi, S; Carta, Gianfranca; Madeddu, Camilla; Lecca, Salvatore; Luchicchi, A; Cadeddu, Francesca; Frau, Roberto; Fattore, L; Fadda, Paola; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA; Fratta, Walter; Schilstrom, B; Banni, Sebastiano; De Montis, Mg; Pistis, Marco | THE JOURNAL OF NEUROSCIENCE | - |
NMDA receptors mediate the role of monoamine oxidase A in pathological aggression | 1-Jan-2012 | Godar, Sc; Bortolato, M; Melis, M; Soggiu, A; Roncada, P; Casu, A; Flore, G; Chen, K; Frau, Roberto; Urbani, A; Castelli, MARIA PAOLA; Devoto, Paola; Shih, Jc | SOCIETY FOR NEUROSCIENCE | - |
Inhibition of steroid 5-alpha reductase reduces marble-burying responses in mice | 1-Jan-2012 | Bini, V; Frau, Roberto; Paba, S; Collu, Maria; Castelli, MARIA PAOLA; Devoto, Paola; Bortolato, M. | - | - |
Reversible disruption of pre-pulse inhibition in hypomorphic-inducible and reversible CB1-/- mice | 1-Jan-2012 | Marongiu, Mfranca; Poddie, D; Porcu, S; Manchinu, Mf; Castelli, MARIA PAOLA; Sogos, Valeria; Bini, V; Frau, Roberto; Caredda, E; Collu, Maria; Ristaldi, Ms | PLOS ONE | - |
Anti-Alcohol and Anxiolytic Properties of a New Chemical Entity, GET73. | 1-Jan-2012 | Loche, A; Simonetti, F; Lobina, C; Carai, Ma; Colombo, G; Castelli, MARIA PAOLA; Barone, D; Cacciaglia, R. | FRONTIERS IN PSYCHIATRY | - |
Characterization of COR627 and COR628, Two Novel Positive Allosteric Modulators of the GABAB Receptor. | 1-Jan-2012 | Castelli, MARIA PAOLA; Casu, A; Casti, P; Lobina, C; Carai, Ma; Colombo, G; Solinas, M; Giunta, D; Mugnaini, C; Pasquini, S; Tafi, A; Brogi, S; Gessa, Gl; Corelli, F. | THE JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS | - |
NMDARs mediate the role of monoamine oxidase A in pathological aggression | 1-Jan-2012 | Bortolato, M; Godar, Sc; Melis, Miriam; Soggiu, A; Roncada, P; Casu, A; Flore, G; Chen, K; Frau, Roberto; Urbani, A; Castelli, MARIA PAOLA; Devoto, Paola; Shih, Jc | THE JOURNAL OF NEUROSCIENCE | - |
Localization of steroid 5α-reductase type 2 isozyme in the adult rat brain | 1-Jan-2011 | Casti, A; Casu, A; Casti, P; Frau, Roberto; Bortolato, M; Spiga, Saturnino; Castelli, MARIA PAOLA; Ennas, Mg | - | SfN |
Effects of drugs of abuse on putative rostromedial tegmental neurons, inhibitory afferents to midbrain dopamine cells | 1-Jan-2011 | Lecca, Salvatore; Melis, Miriam; Luchicchi, A; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA; Muntoni A., L; Pistis, Marco | NEUROPSYCHOPHARMACOLOGY | - |
Adolescent exposure to nicotine and/or the cannabinoid agonist CP 55,940 induces gender-dependent long lasting memory impairments and changes in brain nicotinic and CB1 cannabinoid receptors | 1-Jan-2011 | Mateos, B; Borcel, E; Loriga, R; Luesu, W; Bini, V; Llorente, R; Castelli, MARIA PAOLA; Viveros, Mp | JOURNAL OF PSYCHOPHARMACOLOGY | - |
Methamphetamine neurotoxicity increases brain expression and alters behavioral functions of CB(1) cannabinoid receptors | 1-Jan-2010 | Bortolato, M; Frau, Roberto; Bini, V; Luesu, W; Loriga, Roberta; Collu, Maria; Gessa, Gl; Ennas, MARIA GRAZIA; Castelli, MARIA PAOLA | JOURNAL OF PSYCHIATRIC RESEARCH | - |
Changes induced by acute toxic dose (ATD) of methanphetamine (METH) on cannabinoid CB1 receptors: An immunocytochemistry study | 1-Jan-2009 | Luesu, W; Bini, V; Tuveri, B; Loriga, R; Castelli, MARIA PAOLA; Ennas, MARIA GRAZIA | EUROPEAN JOURNAL OF HISTOCHEMISTRY | - |
Persistent increase in CB1 receptor and amnestic effect of cannabinoid by methamphetamine | 1-Jan-2009 | Frau, Roberto; V., Bini; W., Luesu; Loriga, Roberta; Collu, Maria; G. L., Gessa; M. G., Ennas; M., Bortolato; Castelli, MARIA PAOLA | - | Society for Neurosciences |
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