Synthesis of β-sulfinyl cyclobutane carboxylic amides: Via a formal α to β sulphoxide migration process

Ghisu L.;Melis N.;Serusi L.;Luridiana A.;Soddu F.;Secci F.;Caboni P.;Frongia A.
Supervision
2019-01-01

Abstract

An original tandem reaction consisting of a thermal elimination-addition process was developed. Highly substituted β-sulfinyl cyclobutane carboxylic acid derivatives were obtained from isomeric α-sulfinyl derivatives in a single operation in good to high yields and with high trans diastereoselectivity.
2019
CATALYTIC ENANTIOSELECTIVE SYNTHESIS; DONOR-ACCEPTOR CYCLOBUTANES; CIS/TRANS STEREOCHEMISTRY; AMPHIPHILES INFLUENCE; ASYMMETRIC-SYNTHESIS; SULFENIC ACIDS; DERIVATIVES; INHIBITORS; CYCLOADDITIONS; FOLDAMERS
Files in This Item:
File Size Format  
authorreprints OBC 2019.pdf

Solo gestori archivio

Type: versione editoriale
Size 543.58 kB
Format Adobe PDF
& nbsp; View / Open   Request a copy
543.58 kB Adobe PDF & nbsp; View / Open   Request a copy

Items in DSpace are protected by copyright, with all rights reserved, unless otherwise indicated.

Questionnaire and social

Share on:
Impostazioni cookie