Showing results 1 to 50 of 61
Title Issue Date Author(s) Journal Publisher
Characterization Of The Neurochemical And Behavioral Effects Of The Phenethylamine 2-Cl-4,5-Mdma In Adolescent And Adult Male Rats In press Piras, Gessica; Cadoni, Cristina; Caria, Francesca; Pintori, Nicholas; Spano, Enrica; Vanejevs, Maksims; Ture, Anastasija; Tocco, Graziella; Simola, Nicola; DE LUCA, MARIA ANTONIETTA INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY -
In silico characterization of ligand–receptor interactions for U-47700, N,N-didesmethyl-U-47700, U-50488 at mu- and kappa-opioid receptors 1-Jan-2023 Laus, A; Kumar, A; Caboni, P; DE LUCA, MARIA ANTONIETTA; Baumann, Mh; Pieroni, E; Tocco, G. ARCHIV DER PHARMAZIE -
Dihydroxyphenyl- and Heteroaromatic-Based Thienopyrimidinones to Tackle HIV-1 LEDGF/p75-Dependent IN Activity 1-Jan-2023 Tocco, G.; Canton, S.; Laus, A.; Caboni, P.; Le Grice, S. F. J.; Tramontano, E.; Esposito, F. MOLECULES -
Structural Elucidation of Relevant Gibberellic Acid Impurities and In Silico Investigation of Their Interaction with Soluble Gibberellin Receptor GID1 1-Jan-2023 Caboni, Pierluigi; Laus, Antonio; Eloh, Kodjo; Ntalli, Nikoletta G.; Casula, Mattia; Di Giorgi, Sabrina; Tocco, Graziella ACS OMEGA -
Off‑target activity of NBOMes and NBOMe analogs at the µ opioid receptor 1-Jan-2023 Deventer, Marie H.; Persson, Mattias; Laus, Antonio; Pottie, Eline; Cannaert, Annelies; Tocco, Graziella; Gréen, Henrik; Stove, Christophe P. ARCHIVES OF TOXICOLOGY -
Pharmacological characterization of novel synthetic opioids: Isotonitazene, metonitazene, and piperidylthiambutene as potent μ-opioid receptor agonists 1-Jan-2022 De Luca, Maria Antonietta; Tocco, Graziella; Mostallino, Rafaela; Laus, Antonio; Caria, Francesca; Musa, Aurora; Pintori, Nicholas; Ucha, Marcos; Poza, Celia; Ambrosio, Emilio; Di Chiara, Gaetano; Castelli, M Paola NEUROPHARMACOLOGY -
Mukaiyama reagent: An efficient reaction mediator for rapid synthesis of 1,2-disubstituted-1H-benzo[d]imidazoles 1-Jan-2022 Tocco, G.; Laus, A.; Caboni, P. TETRAHEDRON LETTERS -
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists 1-Jan-2022 Tocco, Graziella; Laus, Antonio; Vanejevs, Maksims; Ture, Anastasija; Mostallino, Rafaela; Pintori, Nicholas; De Luca, Maria Antonietta; Castelli, M. Paola; Di Chiara, Gaetano ARCHIV DER PHARMAZIE -
Electron-Deficient Alkynes as Powerful Tools against Root-Knot Nematode Melodogyne incognita: Nematicidal Activity and Investigation on the Mode of Action 1-Jan-2020 Tocco, Graziella; Eloh, Kodjo; Laus, Antonio; Sasanelli, Nicola; Caboni, Pierluigi JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Scaffold hopping and optimisation of 3’,4’-dihydroxyphenyl- containing thienopyrimidinones: synthesis of quinazolinone derivatives as novel allosteric inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H 1-Jan-2020 Tocco, Graziella; Esposito, Francesca; Caboni, Pierluigi; Laus, Antonio; Beutler, John A.; Wilson, Jennifer A.; Corona, Angela; Le Grice, Stuart F. J.; Tramontano, Enzo JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY -
U-47700 and its analogs: non-fentanyl synthetic opioids impacting the recreational drug market 1-Jan-2020 Baumann, Michael H.; Tocco, Graziella; Papsun, Donna M.; Mohr, Amanda L.; Fogarty, Melissa F.; Krotulski, Alex J. BRAIN SCIENCES -
Uvaria angolensis as a promising source of inhibitors of HIV-1 RT-associated RNA-dependent DNA polymerase and RNase H functions 1-Jan-2018 NGOUTANE MFOPA, Alvine; Corona, Angela; Eloh, Kodjo; Tramontano, Enzo; Frau, Aldo; Boyom, Fabrice Fekam; Caboni, Pierluigi; Tocco, Graziella NATURAL PRODUCT RESEARCH -
Haloacetophenones as newly potent nematicides against Meloidogyne incognita 1-Jan-2017 Tocco, Graziella; Eloh, Kodjo; Onnis, Valentina; Sasanelli, Nicola; Caboni, Pierluigi INDUSTRIAL CROPS AND PRODUCTS -
Solvent-Free addition of indole to aldehydes: Unexpected synthesis of novel 1-[1-(1h-indol-3-yl) alkyl]-1h-indoles and preliminary evaluation of their cytotoxicity in hepatocarcinoma cells 1-Jan-2017 Tocco, Graziella; Zedda, Gloria; Casu, Mariano; Simbula, Gabriella; Begala, Michela MOLECULES -
Nematicidal activity of the volatilome of Eruca sativa on Meloidogyne incognita 1-Jan-2015 Aissani, Nadhem; Urgeghe, Pp; Oplos, C; Saba, M; Tocco, Graziella; Petretto, Gl; Eloh, Kodjo; Menkissoglu Spiroudi, U; Ntalli, Nikoletta; Caboni, Pierluigi JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Tulipaline A: Structure–activity aspects as a nematicide and V-ATPase inhibitor 1-Jan-2014 Caboni, Pierluigi; Tronci, L; Liori, B; Tocco, Graziella; Sasanelli, N; Diana, Andrea PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY -
ZnO-mediated regioselective C-arylsulfonylation of indoles: A facile solvent-free synthesis of 2- and 3-sulfonylindoles and preliminary evaluation of their activity against drug-resistant mutant HIV-1 reverse transcriptases (RTs) 1-Jan-2013 Tocco, Graziella; Begala, Michela; Esposito, Francesca; Caboni, Pierluigi; Cannas, Valeria; Tramontano, Enzo TETRAHEDRON LETTERS -
Active site and allosteric inhibitors of the ribonuclease H activity of HIV reverse transcriptase 1-Jan-2013 Corona, Angela; Masaoka, T; Tocco, Graziella; Tramontano, Enzo; Le Grice, Sfj FUTURE MEDICINAL CHEMISTRY -
Porous silica as host for PEG-supported coumarin molecules 1-Jan-2013 Carbonaro, CARLO MARIA; Casula, MARIA FRANCESCA; Ricci, PIER CARLO; Cubeddu, M; Tocco, Graziella JOURNAL OF MATERIALS SCIENCE -
Potent nematicidal activity of phthalaldehyde, salicylaldehyde, and cinnamic aldehyde against Meloidogyne incognita 1-Jan-2013 Caboni, Pierluigi; Aissani, Nadhem; Cabras, Tiziana; Falqui, Andrea; Marotta, R; Liori, B; Ntalli, Nikoletta; Sarais, Giorgia; Sasanelli, N; Tocco, Graziella JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Nematicidal activity of mint aqueous extracts against the root-knot nematode Meloidogyne incognita 1-Jan-2013 Caboni, Pierluigi; Saba, M; Tocco, Graziella; Casu, Laura; Murgia, A; Maxia, Andrea; Menkissoglu Spiroudi, U; Ntalli, Nikoletta JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Exploiting drug-resistant enzymes as tools to identify thienopyrimidinone inhibitors of human immunodeficiency virus reverse transcriptase-associated ribonuclease H 1-Jan-2013 Masaoka, T; Chung, S; Caboni, Pierluigi; Rausch, Jw; Wilson, Ja; Taskent Sezgin, H; Beutler, Ja; Tocco, Graziella; Le Grice, Sfj JOURNAL OF MEDICINAL CHEMISTRY -
Optical characterization of PEG-supported 7-hydroxy-4-methyl-coumarin in distilled water solution 1-Jan-2012 Carbonaro, CARLO MARIA; Ricci, PIER CARLO; Casula, MARIA FRANCESCA; Tocco, Graziella; Cubeddu, M. JOURNAL OF PHYSICAL CHEMISTRY. A, MOLECULES, SPECTROSCOPY, KINETICS, ENVIRONMENT, & GENERAL THEORY -
Mild Synthetic Approach to Novel Indole-1-Carbinols and Preliminary Evaluation of Their Cytotoxicity in Hepatocarcinoma Cells 1-Jan-2012 Zedda, G; Simbula, G; Begala, M; Pibiri, M; Floris, C; Casu, M; Casu, L; Tocco, G ARCHIV DER PHARMAZIE -
Nematicidal activity of 2-thiophenecarboxaldehyde and methylisothiocyanate from caper (Capparis spinosa) against Meloidogyne incognita 1-Jan-2012 Caboni, Pierluigi; Sarais, Giorgia; Aissani, Nadhem; Tocco, Graziella; Sasanelli, N; Liori, B; Carta, Annarosa; Angioni, Alberto JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY -
Gas-phase ion-molecule reaction of alpha-phenylvinyl cation towards substituted benzenes in the enviroment of an ITMS 1-Jan-2011 Begala, Michela; Tocco, Graziella JOURNAL OF MASS SPECTROMETRY -
Formation of 2-substituted benzofuran fragment ions from 6-alkyl- and 6-aryldibenzo(d,f)(1,3)dioxepine derivatives under electron ionization-a useful precursor ion for isomeric differentiation. 1-Jan-2009 Begala, Michela; Tocco, Graziella; Meli, G; Podda, G; Urru, Sa - -
Evaluation of Photoluminescence Properties of Some Poly(ethylene glycol) – Supported Coumarin Derivatives 1-Jan-2009 Tocco, Graziella; Carbonaro, CARLO MARIA; Meli, G; Podda, G. MOLECULES -
PEG-immobilization of cardol and soluble polymer-supported synthesis of some cardol–coumarin derivatives: Preliminary evaluation of their inhibitory activity on mushroom tyrosinase 1-Jan-2009 Tocco, Graziella; Fais, Antonella; Meli, G; Begala, Michela; Podda, G; FADDA M., B; Corda, M; ATTANASI O., A; Filippone, P; Berretta, S. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS -
InCl3 and ZrCl4 catalyzed regioselective reaction of 2,2'-dihydroxybiphenyl with terminal alkynes: synthesis of new dibenzo[d,f][1,3]dioxepines 1-Jan-2008 Tocco, Graziella; Begala, Michela; Meli, G; Podda, G. TETRAHEDRON -
Chemoselective synthesis of new dibenzo[d,f]-1,3-dioxepines and 12H-dibenzo[d,g]-1,3-dioxocines 1-Jan-2007 Tocco, Graziella; Begala, Michela; Meli, G; Podda, G. HETEROCYCLES -
2-Substituted benzofuran fragment ion formation in the electron ionization mass spectra of 6-alkyl- and 6-aryldibenzo(d,f)-(1,3)dioxepine derivatives.1. Spirocyclization of the molecular ions in the gas phase 1-Jan-2007 Begala, Michela; Tocco, Graziella; Meli, G; Podda, G; URRU AM, S. RAPID COMMUNICATIONS IN MASS SPECTROMETRY -
Electron ionization-induced fragmentation of some new dibenzo (d,f)(1,3) dioxepine derivatives 1-Jan-2006 Begala, Michela; Tocco, Graziella; Delogu, GIOVANNA LUCIA; Meli, G; Picciau, MARIA CARMEN; Podda, G. JOURNAL OF MASS SPECTROMETRY -
SINTESI E IMMOBILIZZAZIONE DI ALCUNE CUMARINE ANALOGHE DEL RESVERATROLO AL POLIETILENGLICOLE 1-Jan-2006 Begala, Michela; Delogu, GIOVANNA LUCIA; G., Meli; C., Picciau; G., Podda; Tocco, Graziella; S., Urru - -
Sintesi e Caratterizzazione Strutturale di Derivati Cumarinici Contenenti Gruppi 1,3-Diossolici 1-Jan-2005 Delogu, GIOVANNA LUCIA; Begala, Michela; Picciau, MARIA CARMEN; Podda, G; Tocco, Graziella - -
SINTESI E CARATTERIZZAZIONE STRUTTURALE DI DERIVATI CUMARINICI CONTENETI GRUPPI 1,3-DIOSSOLICI 1-Jan-2005 Delogu, GIOVANNA LUCIA; Begala, Michela; G., Meli; C., Picciau; G., Podda; Tocco, Graziella - -
SINTESI ONE-STEP InCl3-CATALIZZATA DI NUOVI DERIVATI DELLE DIBENZO(D,F)(1,3)DIOXEPINE E 12H-DIBENZO(D,G)(1,3)DIOXACINE A PARTIRE DA SUBSTRATI ALDEIDICI ED ACETILENICI 1-Jan-2005 Tocco, Graziella; Begala, Michela; Delogu, GIOVANNA LUCIA; G., Mel; . C., Picciau; G., Podda - -
CHARACTERISATION OF DIBENZO(d,f)(1,3)DIOXEPINE DERIVATIVES BY MULTIPLE STAGE MASS SPECTROMETRY 1-Jan-2005 Begala, Michela; Tocco, Graziella; Delogu, GIOVANNA LUCIA; G., Meli; C., Picciau; G., Podda - -
Soluble Polymer-Supported Synthesis of 4-Methyl Coumarin on Modified Poly(ethylene glycol)s 1-Jan-2005 Tocco, Graziella; Begala, Michela; Delogu, GIOVANNA LUCIA; Meli, G; Picciau, MARIA CARMEN; Podda, G. SYNLETT -
Characterisation of new pyridazinofurocoumarins by electron ionisation and multiple stage tandem mass spectrometry using an ion trap mass spectrometer 1-Jan-2004 Begala, Michela; GONZALEZ GOMEZ, J. C.; Podda, G; Santana, L.; Tocco, Graziella; Uriarte, E. RAPID COMMUNICATIONS IN MASS SPECTROMETRY -
A New Synthesis of 1,3,5-Triazine with Coumarin Derivatives”e “Synthesis and Immobilization of Some Coumarine Derivatives on a Modified Poly(ethylene glycol 1-Jan-2004 Tocco, Graziella; Begala, Michela - -
IMMOBILIZZAZIONE E SINTESI IN FASE LIQUIDA PEG-SUPPORTATA DI ALCUNI DERIVATI CUMARINICI 1-Jan-2004 Tocco, Graziella; Begala, Michela; Delogu, GIOVANNA LUCIA; C., Picciau; G., Podda - -
Impiego dell'indio (III) cloruro come catalizzatore nella sintesi one-step di nuovi derivati delle dibenzo(d,f)(1,3)dioxepine e 12H-dibenzo(d,g)(1,3)dioxacine 1-Jan-2004 Tocco, Graziella; Begala, Michela; Delogu, GIOVANNA LUCIA; C., Picciau; G., Podda - -
Sintesi e caratterizzazione di una nuova classe di derivati cumarinici con 1,3,5-triazina 1-Jan-2004 Begala, Michela; Delogu, GIOVANNA LUCIA; Picciau, MARIA CARMEN; G., Podda; Tocco, Graziella; E., Quezada; L., Santana; E., Uriarte - -
An efficient and direct route to obtain 4’-(Furocoumarin)acetates 1-Jan-2004 Begala, Michela; Delogu, GIOVANNA LUCIA; Picciau, MARIA CARMEN; Podda, G; Tocco, Graziella; Quezada, E; Santana, L; Uriarte, E. - -
Via diretta per sintetizzare 4’-( furocumarine) acetato 1-Jan-2004 Begala, Michela; Delogu, GIOVANNA LUCIA; Picciau, MARIA CARMEN; G., Podda; Tocco, Graziella; E., Quezada; L., Santana; E., Uriarte - -
5th Spanish Italian Symposium on Organic Chemistry 1-Jan-2004 Begala, Michela; Delogu, GIOVANNA LUCIA; C., Picciau; G., Podda; Tocco, Graziella; E., Quezada; E., Uriarte - -
Indium(III) chloride catalyzed one step synthesis of some new dibenzo(d,f)(1,3)dioxepines and 12H-dibenzo(d,g)(1,3)dioxocin derivatives 1-Jan-2004 Tocco, Graziella; Begala, Michela; Delogu, GIOVANNA LUCIA; Picciau, MARIA CARMEN; Podda, G. TETRAHEDRON LETTERS -
SINTESI E CARATTERIZZAZIONE DI PIRIDAZINO FUROCUMARINE 1-Jan-2003 Delogu, GIOVANNA LUCIA; Begala, M; Gomez, Jc; Podda, G; Santana, L; Tocco, Graziella; Uriarte, E. - -
Synthesis and Application of New Fluorescent Phase Transfer Catalysts Based on Crown Coumarin Structure 1-Jan-2003 Delogu, GIOVANNA LUCIA; Picciau, MARIA CARMEN; Tocco, Graziella; Santana, L; Uriarte, E. - -
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