University of Cagliari
Roberta Loddo
Design, synthesis, and antiviral activities of new benzotriazole-based derivatives
2023-01-01 Ibba, R.; Corona, P.; Nonne, F.; Caria, P.; Serreli, G.; Palmas, V.; Riu, F.; Sestito, S.; Nieddu, M.; Loddo, R.; Sanna, G.; Sandra Piras, S.
Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication
2022-01-01 Ibba, Roberta; Riu, Federico; Delogu, Ilenia; Lupinu, Ilenia; Carboni, Gavino; Loddo, Roberta; Piras, Sandra; Carta, Antonio
Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives
2021-01-01 Ibba, R.; Piras, S.; Corona, P.; Riu, F.; Loddo, R.; Delogu, I.; Collu, G.; Sanna, G.; Caria, P.; Dettori, T.; Carta, A.
Inhibition of enterovirus a71 by a novel 2-phenyl-benzimidazole derivative
2021-01-01 Ibba, R.; Carta, A.; Madeddu, S.; Caria, P.; Serreli, G.; Piras, S.; Sestito, S.; Loddo, R.; Sanna, G.
Anti-BVDV activity evaluation of naphthoimidazole derivatives compared with parental imidazoquinoline compounds.
2020-01-01 Ibba, R.; Piras, S.; Delogu, I.; Loddo, R.; Carta, A.
Preliminary anti-Coxsackie activity of novel 1-[4-(5,6-dimethyl(H)-1H(2H)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas
2020-01-01 Piras, S.; Corona, P.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A.
Antiviral activity of benzotriazole based derivatives
2020-01-01 Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A.
5,6-Dichloro-2-phenyl-benzotriazoles: New potent inhibitors of orthohantavirus
2020-01-01 Sanna, G.; Piras, S.; Madeddu, S.; Busonera, B.; Klempa, B.; Corona, P.; Ibba, R.; Murineddu, G.; Carta, A.; Loddo, R.
Dichloro-phenyl-benzotriazoles: a new selective class of human respiratory syncytial virus entry inhibitors
2019-01-01 Piras, S.; Sanna, G.; Carta, A.; Corona, P.; Ibba, R.; Loddo, R.; Madeddu, S.; Caria, P.; Aulic, S.; Laurini, E.; Fermeglia, M.; and Pricl, S
Design, synthesis, antiviral evaluation, and SAR studies of new 1-(phenylsulfonyl)-1H-pyrazol -4-yl-methylaniline derivatives.
2019-01-01 Desideri, N.; Fioravanti, R.; Proietti Monaco, L.; Atzori, E. M.; Carta, A.; Delogu, I.; Collu, G.; and Loddo, R
9-Aminoacridine-based agents impair the bovine viral diarrhea virus (BVDV) replication targeting the RNA-dependent RNA polymerase (RdRp)
2018-01-01 Loddo, R.; Francesconi, V.; Laurini, E.; Boccardo, S.; Aulic, S.; Fermeglia, M.; Pricl, S.; Tonelli, M.
Benzimidazole derivatives endowed with potent antileishmanial activity
2018-01-01 Tonelli, M.; Gabriele, E.; Piazza, F.; Basilico, N.; Parapini, S.; Tasso, B.; Loddo, R.; Sparatore, F.; Sparatore, A.
Antiviral activities of 5-chlorobenzotriazole derivatives
2018-01-01 Ibba, R.; Corona, P.; Carta, A.; Giunchedi, P.; Loddo, R.; Sanna, G.; Delogu, I.; Piras, S.
Quinoxaline derivatives as new inhibitors of coxsackievirus B5
2018-01-01 Carta, A.; Sanna, G.; Briguglio, I.; Madeddu, S.; Vitale, G.; Piras, S.; Corona, P.; Peana, A. T.; Laurini, E.; Fermeglia, M.; Pricl, S.; Serra, A.; Carta, Elisa; Loddo, R.; Giliberti, G.
Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles
2017-01-01 Cichero, E.; Tonelli, M.; Novelli, F.; Tasso, B.; Delogu, Ilenia; Loddo, Roberta; Bruno, O.; Fossa, P.
Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus
2017-01-01 Tonelli, M; Naesens, L; Gazzarrini, S; Santucci, M; Cichero, E; Tasso, B; Moroni, A; Costi, Mp; Loddo, Roberta
Synthesis, structural characterization and biological evaluation of 4'-C-methyl- and phenyl-dioxolane pyrimidine and purine nucleosides
2017-01-01 Franchisi, S.; Battisti, U. m.; Sorbi, C.; Tait, A.; Cornia, A.; Jeong, L. s.; Lee, S. k.; Song, J.; Loddo, Roberta; Madeddu, Silvia; Sanna, Giuseppina; Brasili, L.
Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation.
2017-01-01 Fioravanti, R.; Desideri, N.; Carta, A.; Atzori E., M.; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta
Facile synthesis of the NNRTI microbicide MC-1220 and synthesis of its phosphoramidate prodrugs
2016-01-01 Loksha, Ym; Pedersen, Eb; LA COLLA, Paolo; Loddo, Roberta
Activity of bis(7-hydroxycoumarin) Mannich bases against bovine viral diarrhoea virus
2016-01-01 Ibrahim, M. M.; Mazzei, M.; Delogu, Ilenia; Szabo, Robert; Sanna, Giuseppina; Loddo, Roberta
Synthesis and antiviral evaluation of 1-[(2-Phenoxyethyl)oxymethyl] and 6-(3,5-Dimethoxybenzyl) analogues of HIV drugs emivirine and TNK-651
2016-01-01 El Brollosy, Nr; Loddo, Roberta
Synthesis and anti-HIV-1 evaluation of some novel MC-1220 analogs as non-nucleoside reverse transcriptase inhibitors
2016-01-01 Loksha, Ym; Pedersen, Eb; Loddo, Roberta; LA COLLA, Paolo
A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems
2016-01-01 Carta, A; Briguglio, I; Piras, S; Corona, P; Ibba, R; Laurini, E; Fermeglia, M; Pricl, S; Desideri, N; Atzori, Em; La Colla, P; Collu, G; Delogu, I; Loddo, R
Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5
2015-01-01 Loddo, Roberta; Novelli, F; Sparatore, A; Tasso, B; Tonelli, M; Boido, V; Sparatore, F; Collu, Gabriella; Delogu, Ilenia; Giliberti, Gabriele; LA COLLA, Paolo
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agents
2015-01-01 Spallarossa, Andrea; Caneva, Chiara; Caviglia, Matteo; Alfei, Silvana; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Brindisi, Margherita; Zisterer, Daniela M.; Bright, Sandra A.; Williams, Clive D.; Crespan, Emmanuele; Maga, Giovanni; Sanna, Giuseppina; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives
2015-01-01 Briguglio, I; Loddo, Roberta; Laurini, E; Fermeglia, M; Piras, S; Corona, P; Giunchedi, P; Gavini, E; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; LA COLLA, Paolo; Pricl, S; Carta, A.
Synthesis and biological evaluation of (acyl)hydrazones and thiosemicarbazones obtained via in situ condensation of iminium salts with nitrogen-containing nucleophiles.
2015-01-01 Caneva, C; Alfei, S; De Maria, M; Ibba, Cristina; Delogu, Ilenia; Spallarossa, A; Loddo, Roberta
N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents
2015-01-01 Fioravanti, R; Desideri, N; Biava, M; Droghini, P; Atzori, Em; Ibba, Cristina; Collu, Gabriella; Sanna, Giuseppina; Delogu, Ilenia; Loddo, Roberta
Synthesis of novel fluoro analogues of MKC442 as microbicides
2014-01-01 Loksha, Ym; Pedersen, Eb; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Giliberti, Gabriele; La Colla, P.
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines
2014-01-01 Loddo, Roberta; Briguglio, I; Corona, P; Piras, S; Loriga, M; Paglietti, G; Carta, A; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, P; La Colla, P.
Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines.
2014-01-01 Tonelli, M; Novelli, F; Tasso, B; Sparatore, A; Boido, V; Sparatore, F; Cannas, S; Molicotti, P; Zanetti, S; Parapini, S; Loddo, Roberta
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
2014-01-01 Tonelli, M; Novelli, F; Tasso, B; Vazzana, I; Sparatore, A; Boido, V; Sparatore, F; La Colla, P; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, B; Farci, P; Ibba, Cristina; Loddo, Roberta
Erratum to: Syntheses and in vitro biological screening of 1-aryl-10 H-[1,2,4]triazolo[3′,4′:3,4][1,2,4]triazino[5,6-b]indoles
2013-01-01 Upadhyay, K; Manvar, A; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A; Giliberti, Gabriele; Secci, B; Busonera, B; Sanna, Giuseppina; Loddo, Roberta; La Colla, P.
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents
2013-01-01 Spallarossa, A; Rotolo, C; Sissi, C; Marson, G; Greco, Ml; Ranise, A; La Colla, P; Busonera, B; Loddo, Roberta
Syntheses and in vitro biologic screening 3 of 1-aryl-10H-[1,2,4]triazolo[30,40:3,4][1,2,4]triazino[5,6-b]indoles
2013-01-01 Upadhyay, K; Manvar, A; Loddo, Roberta; La Colla, P; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A.
A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220
2012-01-01 Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, Roberta; La Colla, P.
Synthesis and biological evaluation of new 3-phenyl-1-[(4-arylpiperazin-1-yl)alkyl]-piperidine-2,6-diones
2011-01-01 Bielenica, A; Kossakowski, J; Struga, M; Dybala, I; Loddo, Roberta; Ibba, Cristina; La Colla, P.
Biological evaluation of novel 1,4-dithiine derivatives as potential antimicrobial agents
2011-01-01 Bielenica, A; Kossakowski, J; Struga, M; Dybała, I; La Colla, P; Tamburini, Elena; Loddo, Roberta
3-Aryl-2-[1H-benzotriazol-1-yl]acrylonitriles: a novel class of potent tubulin inhibitors
2011-01-01 Carta, A.; Briguglio, I.; Piras, S.; Boatto, G.; La Colla, P.; Loddo, R.; Tolomeo, M.; Grimaudo, S.; Di Cristina, A.; Pipitone, R. M.; Laurini, E.; Paneni, M. S.; Posocco, P.; Fermeglia, M.; and Pricl, S.
Synthesis and anti-HIV-1 activity of new fluoro-HEPT analogues: an investigation on fluoro versus hydroxy substituents
2011-01-01 Loksha, Ym; Pedersen, Eb; Loddo, Roberta; LA COLLA, P.
Topical nonnucleoside reverse transcriptase inhibitor MC 1220 partially prevents vaginal RT-SHIV infection of macaques
2011-01-01 Stolte Leeb, N.; Loddo, Roberta; Antimisiaris, S.; Schultheiss, T.; Sauermann, U.; Franz, M.; Mourtas, S.; Parsy, C.; Storer, R.; LA COLLA, Paolo; Stahl Hennig, C.
Synthesis and in vitro anti-HIV activity of N-1,3-benzo[d]thiazol-2-yl-2-(2-oxo-2H-chromen-4-yl)acetamide derivatives using MTT method
2011-01-01 Bhavsar, D; Trivedi, J; Parekh, S; Savant, M; Thakrar, S; Bavishi, A; Radadiya, A; Vala, H; Lunagariya, J; Parmar, M; Paresh, L; Loddo, Roberta; Shah, A.
2,3-dihydro-1,2-diphenyl-substituted 4H-pyridinone derivatives as new anti flaviviridae inhibitors
2011-01-01 Peduto, A; Massa, A; DI MOLA, A; DE CAPRARIIS, P; LA COLLA, P; Loddo, Roberta; Altamura, S; Maga, G; Filosa, R.
1,2-benzisothiazol-3(2h)-one benzenesulfonamides targeting the hiv nucleocapsid proteins are potential microbicide candidates for the prevention of mucosal hiv transmission/acquisition
2010-01-01 Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; Giliberti, Gabriele; Marongiu, E.; Loddo, Roberta; La Colla, P.
Platinum and palladium-triazole complexes as highly potential antitumor agents
2010-01-01 AL MASOUDI, Na; Abdullah, Bh; Essa, Ah; Loddo, Roberta; AND LA COLLA, P.
A novel synthetic route for the anti-HIV drug MC-1220 and its analogues
2010-01-01 Loksha, Ym; Globisch, D; Loddo, Roberta; Collu, G; LA COLLA, P; Pedersen, Eb
Styrylbenzimidazoles. Synthesis and biological activity - part 3
2010-01-01 Vitale, G; Corona, P; Loriga, M; Loddo, Roberta; Paglietti, G; Ibba, Cristina; Giliberti, Gabriele; Loddo, R; Marongiu, E; La Colla, P.
Antiviral activity of benzimidazole derivatives. II. Antiviral activity of 2-phenylbenzimidazole derivatives
2010-01-01 Tonelli, M; Simone, M; Tasso, B; Novelli, F; Boido, V; Sparatore, F; Paglietti, G; Pricl, S; Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Ibba, Cristina; Sanna, Giuseppina; Loddo, Roberta; La Colla, P.
Synthesis, in vitro antiproliferative and anti-HIV activity of new derivatives of 2-Piperazino-1,3-benzo[d]thiazoles
2010-01-01 AL SOUD, Ya; AL SA'DONI, Hh; Saber, Sow; AL SHANEEK, Rhm; AL MASOUDI, Na; Loddo, Roberta; LA COLLA, P.
Protective properties of non-nucleoside reverse transcriptase inhibitor (MC1220) incorporated into liposome against intravaginal challenge of Rhesus Macaques with RT-SHIV
2010-01-01 Caron, M; Besson, G; Etenna, Sl; MINTSA NDONG, A; Mourtas, S; Radaelli, A; Morghen, Cd; Loddo, Roberta; LA COLLA, P; Antimisiaris, Sg; Kazanji, M.
| Title | Issue Date | Author(s) | Journal | Publisher |
|---|---|---|---|---|
| Design, synthesis, and antiviral activities of new benzotriazole-based derivatives | 1-Jan-2023 | Ibba, R.; Corona, P.; Nonne, F.; Caria, P.; Serreli, G.; Palmas, V.; Riu, F.; Sestito, S.; Nieddu, M.; Loddo, R.; Sanna, G.; Sandra Piras, S. | PHARMACEUTICALS | - |
| Benzimidazole-2-Phenyl-Carboxamides as Dual-Target Inhibitors of BVDV Entry and Replication | 1-Jan-2022 | Ibba, Roberta; Riu, Federico; Delogu, Ilenia; Lupinu, Ilenia; Carboni, Gavino; Loddo, Roberta; Piras, Sandra; Carta, Antonio | VIRUSES | - |
| Synthesis, Antitumor and Antiviral In Vitro Activities of New Benzotriazole-Dicarboxamide Derivatives | 1-Jan-2021 | Ibba, R.; Piras, S.; Corona, P.; Riu, F.; Loddo, R.; Delogu, I.; Collu, G.; Sanna, G.; Caria, P.; Dettori, T.; Carta, A. | FRONTIERS IN CHEMISTRY | - |
| Inhibition of enterovirus a71 by a novel 2-phenyl-benzimidazole derivative | 1-Jan-2021 | Ibba, R.; Carta, A.; Madeddu, S.; Caria, P.; Serreli, G.; Piras, S.; Sestito, S.; Loddo, R.; Sanna, G. | VIRUSES | - |
| Anti-BVDV activity evaluation of naphthoimidazole derivatives compared with parental imidazoquinoline compounds. | 1-Jan-2020 | Ibba, R.; Piras, S.; Delogu, I.; Loddo, R.; Carta, A. | THE OPEN MEDICINAL CHEMISTRY JOURNAL | - |
| Preliminary anti-Coxsackie activity of novel 1-[4-(5,6-dimethyl(H)-1H(2H)-benzotriazol-1(2)-yl)phenyl]-3-alkyl(aryl)ureas | 1-Jan-2020 | Piras, S.; Corona, P.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A. | MEDICINAL CHEMISTRY | - |
| Antiviral activity of benzotriazole based derivatives | 1-Jan-2020 | Corona, P.; Piras, S.; Ibba, R.; Riu, F.; Murineddu, G.; Sanna, G.; Madeddu, S.; Delogu, I.; Loddo, R.; Carta, A. | THE OPEN MEDICINAL CHEMISTRY JOURNAL | - |
| 5,6-Dichloro-2-phenyl-benzotriazoles: New potent inhibitors of orthohantavirus | 1-Jan-2020 | Sanna, G.; Piras, S.; Madeddu, S.; Busonera, B.; Klempa, B.; Corona, P.; Ibba, R.; Murineddu, G.; Carta, A.; Loddo, R. | VIRUSES | - |
| Dichloro-phenyl-benzotriazoles: a new selective class of human respiratory syncytial virus entry inhibitors | 1-Jan-2019 | Piras, S.; Sanna, G.; Carta, A.; Corona, P.; Ibba, R.; Loddo, R.; Madeddu, S.; Caria, P.; Aulic, S.; Laurini, E.; Fermeglia, M.; and Pricl, S | FRONTIERS IN CHEMISTRY | - |
| Design, synthesis, antiviral evaluation, and SAR studies of new 1-(phenylsulfonyl)-1H-pyrazol -4-yl-methylaniline derivatives. | 1-Jan-2019 | Desideri, N.; Fioravanti, R.; Proietti Monaco, L.; Atzori, E. M.; Carta, A.; Delogu, I.; Collu, G.; and Loddo, R | FRONTIERS IN CHEMISTRY | - |
| 9-Aminoacridine-based agents impair the bovine viral diarrhea virus (BVDV) replication targeting the RNA-dependent RNA polymerase (RdRp) | 1-Jan-2018 | Loddo, R.; Francesconi, V.; Laurini, E.; Boccardo, S.; Aulic, S.; Fermeglia, M.; Pricl, S.; Tonelli, M. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Benzimidazole derivatives endowed with potent antileishmanial activity | 1-Jan-2018 | Tonelli, M.; Gabriele, E.; Piazza, F.; Basilico, N.; Parapini, S.; Tasso, B.; Loddo, R.; Sparatore, F.; Sparatore, A. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Antiviral activities of 5-chlorobenzotriazole derivatives | 1-Jan-2018 | Ibba, R.; Corona, P.; Carta, A.; Giunchedi, P.; Loddo, R.; Sanna, G.; Delogu, I.; Piras, S. | MONATSHEFTE FÜR CHEMIE | - |
| Quinoxaline derivatives as new inhibitors of coxsackievirus B5 | 1-Jan-2018 | Carta, A.; Sanna, G.; Briguglio, I.; Madeddu, S.; Vitale, G.; Piras, S.; Corona, P.; Peana, A. T.; Laurini, E.; Fermeglia, M.; Pricl, S.; Serra, A.; Carta, Elisa; Loddo, R.; Giliberti, G. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles | 1-Jan-2017 | Cichero, E.; Tonelli, M.; Novelli, F.; Tasso, B.; Delogu, Ilenia; Loddo, Roberta; Bruno, O.; Fossa, P. | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | - |
| Host dihydrofolate reductase (DHFR)-directed cycloguanil analogues endowed with activity against influenza virus and respiratory syncytial virus | 1-Jan-2017 | Tonelli, M; Naesens, L; Gazzarrini, S; Santucci, M; Cichero, E; Tasso, B; Moroni, A; Costi, Mp; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis, structural characterization and biological evaluation of 4'-C-methyl- and phenyl-dioxolane pyrimidine and purine nucleosides | 1-Jan-2017 | Franchisi, S.; Battisti, U. m.; Sorbi, C.; Tait, A.; Cornia, A.; Jeong, L. s.; Lee, S. k.; Song, J.; Loddo, Roberta; Madeddu, Silvia; Sanna, Giuseppina; Brasili, L. | ARCHIVES OF PHARMACAL RESEARCH | - |
| Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation. | 1-Jan-2017 | Fioravanti, R.; Desideri, N.; Carta, A.; Atzori E., M.; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Facile synthesis of the NNRTI microbicide MC-1220 and synthesis of its phosphoramidate prodrugs | 1-Jan-2016 | Loksha, Ym; Pedersen, Eb; LA COLLA, Paolo; Loddo, Roberta | ORGANIC & BIOMOLECULAR CHEMISTRY | - |
| Activity of bis(7-hydroxycoumarin) Mannich bases against bovine viral diarrhoea virus | 1-Jan-2016 | Ibrahim, M. M.; Mazzei, M.; Delogu, Ilenia; Szabo, Robert; Sanna, Giuseppina; Loddo, Roberta | ANTIVIRAL RESEARCH | - |
| Synthesis and antiviral evaluation of 1-[(2-Phenoxyethyl)oxymethyl] and 6-(3,5-Dimethoxybenzyl) analogues of HIV drugs emivirine and TNK-651 | 1-Jan-2016 | El Brollosy, Nr; Loddo, Roberta | DRUG RESEARCH | - |
| Synthesis and anti-HIV-1 evaluation of some novel MC-1220 analogs as non-nucleoside reverse transcriptase inhibitors | 1-Jan-2016 | Loksha, Ym; Pedersen, Eb; Loddo, Roberta; LA COLLA, Paolo | ARCHIV DER PHARMAZIE | - |
| A combined in silico/in vitro approach unveils common molecular requirements for efficient BVDV RdRp binding of linear aromatic N-polycyclic systems | 1-Jan-2016 | Carta, A; Briguglio, I; Piras, S; Corona, P; Ibba, R; Laurini, E; Fermeglia, M; Pricl, S; Desideri, N; Atzori, Em; La Colla, P; Collu, G; Delogu, I; Loddo, R | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Antiviral activity of benzotriazole derivatives. 5-[4-(Benzotriazol-2-yl)phenoxy]-2,2-dimethylpentanoic acids potently and selectively inhibit Coxsackie Virus B5 | 1-Jan-2015 | Loddo, Roberta; Novelli, F; Sparatore, A; Tasso, B; Tonelli, M; Boido, V; Sparatore, F; Collu, Gabriella; Delogu, Ilenia; Giliberti, Gabriele; LA COLLA, Paolo | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agents | 1-Jan-2015 | Spallarossa, Andrea; Caneva, Chiara; Caviglia, Matteo; Alfei, Silvana; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Brindisi, Margherita; Zisterer, Daniela M.; Bright, Sandra A.; Williams, Clive D.; Crespan, Emmanuele; Maga, Giovanni; Sanna, Giuseppina; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives | 1-Jan-2015 | Briguglio, I; Loddo, Roberta; Laurini, E; Fermeglia, M; Piras, S; Corona, P; Giunchedi, P; Gavini, E; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; LA COLLA, Paolo; Pricl, S; Carta, A. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and biological evaluation of (acyl)hydrazones and thiosemicarbazones obtained via in situ condensation of iminium salts with nitrogen-containing nucleophiles. | 1-Jan-2015 | Caneva, C; Alfei, S; De Maria, M; Ibba, Cristina; Delogu, Ilenia; Spallarossa, A; Loddo, Roberta | MOLECULAR DIVERSITY | - |
| N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents | 1-Jan-2015 | Fioravanti, R; Desideri, N; Biava, M; Droghini, P; Atzori, Em; Ibba, Cristina; Collu, Gabriella; Sanna, Giuseppina; Delogu, Ilenia; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
| Synthesis of novel fluoro analogues of MKC442 as microbicides | 1-Jan-2014 | Loksha, Ym; Pedersen, Eb; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Giliberti, Gabriele; La Colla, P. | JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines | 1-Jan-2014 | Loddo, Roberta; Briguglio, I; Corona, P; Piras, S; Loriga, M; Paglietti, G; Carta, A; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, P; La Colla, P. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Antitubercular activity of quinolizidinyl/pyrrolizidinylalkyliminophenazines. | 1-Jan-2014 | Tonelli, M; Novelli, F; Tasso, B; Sparatore, A; Boido, V; Sparatore, F; Cannas, S; Molicotti, P; Zanetti, S; Parapini, S; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents | 1-Jan-2014 | Tonelli, M; Novelli, F; Tasso, B; Vazzana, I; Sparatore, A; Boido, V; Sparatore, F; La Colla, P; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, B; Farci, P; Ibba, Cristina; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Erratum to: Syntheses and in vitro biological screening of 1-aryl-10 H-[1,2,4]triazolo[3′,4′:3,4][1,2,4]triazino[5,6-b]indoles | 1-Jan-2013 | Upadhyay, K; Manvar, A; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A; Giliberti, Gabriele; Secci, B; Busonera, B; Sanna, Giuseppina; Loddo, Roberta; La Colla, P. | MEDICINAL CHEMISTRY RESEARCH | - |
| Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents | 1-Jan-2013 | Spallarossa, A; Rotolo, C; Sissi, C; Marson, G; Greco, Ml; Ranise, A; La Colla, P; Busonera, B; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Syntheses and in vitro biologic screening 3 of 1-aryl-10H-[1,2,4]triazolo[30,40:3,4][1,2,4]triazino[5,6-b]indoles | 1-Jan-2013 | Upadhyay, K; Manvar, A; Loddo, Roberta; La Colla, P; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A. | MEDICINAL CHEMISTRY RESEARCH | - |
| A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220 | 1-Jan-2012 | Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, Roberta; La Colla, P. | - | - |
| Synthesis and biological evaluation of new 3-phenyl-1-[(4-arylpiperazin-1-yl)alkyl]-piperidine-2,6-diones | 1-Jan-2011 | Bielenica, A; Kossakowski, J; Struga, M; Dybala, I; Loddo, Roberta; Ibba, Cristina; La Colla, P. | SCIENTIA PHARMACEUTICA | - |
| Biological evaluation of novel 1,4-dithiine derivatives as potential antimicrobial agents | 1-Jan-2011 | Bielenica, A; Kossakowski, J; Struga, M; Dybała, I; La Colla, P; Tamburini, Elena; Loddo, Roberta | MEDICINAL CHEMISTRY RESEARCH | - |
| 3-Aryl-2-[1H-benzotriazol-1-yl]acrylonitriles: a novel class of potent tubulin inhibitors | 1-Jan-2011 | Carta, A.; Briguglio, I.; Piras, S.; Boatto, G.; La Colla, P.; Loddo, R.; Tolomeo, M.; Grimaudo, S.; Di Cristina, A.; Pipitone, R. M.; Laurini, E.; Paneni, M. S.; Posocco, P.; Fermeglia, M.; and Pricl, S. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
| Synthesis and anti-HIV-1 activity of new fluoro-HEPT analogues: an investigation on fluoro versus hydroxy substituents | 1-Jan-2011 | Loksha, Ym; Pedersen, Eb; Loddo, Roberta; LA COLLA, P. | ARCHIV DER PHARMAZIE | - |
| Topical nonnucleoside reverse transcriptase inhibitor MC 1220 partially prevents vaginal RT-SHIV infection of macaques | 1-Jan-2011 | Stolte Leeb, N.; Loddo, Roberta; Antimisiaris, S.; Schultheiss, T.; Sauermann, U.; Franz, M.; Mourtas, S.; Parsy, C.; Storer, R.; LA COLLA, Paolo; Stahl Hennig, C. | AIDS RESEARCH AND HUMAN RETROVIRUSES | - |
| Synthesis and in vitro anti-HIV activity of N-1,3-benzo[d]thiazol-2-yl-2-(2-oxo-2H-chromen-4-yl)acetamide derivatives using MTT method | 1-Jan-2011 | Bhavsar, D; Trivedi, J; Parekh, S; Savant, M; Thakrar, S; Bavishi, A; Radadiya, A; Vala, H; Lunagariya, J; Parmar, M; Paresh, L; Loddo, Roberta; Shah, A. | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
| 2,3-dihydro-1,2-diphenyl-substituted 4H-pyridinone derivatives as new anti flaviviridae inhibitors | 1-Jan-2011 | Peduto, A; Massa, A; DI MOLA, A; DE CAPRARIIS, P; LA COLLA, P; Loddo, Roberta; Altamura, S; Maga, G; Filosa, R. | CHEMICAL BIOLOGY & DRUG DESIGN | - |
| 1,2-benzisothiazol-3(2h)-one benzenesulfonamides targeting the hiv nucleocapsid proteins are potential microbicide candidates for the prevention of mucosal hiv transmission/acquisition | 1-Jan-2010 | Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; Giliberti, Gabriele; Marongiu, E.; Loddo, Roberta; La Colla, P. | - | - |
| Platinum and palladium-triazole complexes as highly potential antitumor agents | 1-Jan-2010 | AL MASOUDI, Na; Abdullah, Bh; Essa, Ah; Loddo, Roberta; AND LA COLLA, P. | ARCHIV DER PHARMAZIE | - |
| A novel synthetic route for the anti-HIV drug MC-1220 and its analogues | 1-Jan-2010 | Loksha, Ym; Globisch, D; Loddo, Roberta; Collu, G; LA COLLA, P; Pedersen, Eb | CHEMMEDCHEM | - |
| Styrylbenzimidazoles. Synthesis and biological activity - part 3 | 1-Jan-2010 | Vitale, G; Corona, P; Loriga, M; Loddo, Roberta; Paglietti, G; Ibba, Cristina; Giliberti, Gabriele; Loddo, R; Marongiu, E; La Colla, P. | MEDICINAL CHEMISTRY | - |
| Antiviral activity of benzimidazole derivatives. II. Antiviral activity of 2-phenylbenzimidazole derivatives | 1-Jan-2010 | Tonelli, M; Simone, M; Tasso, B; Novelli, F; Boido, V; Sparatore, F; Paglietti, G; Pricl, S; Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Ibba, Cristina; Sanna, Giuseppina; Loddo, Roberta; La Colla, P. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
| Synthesis, in vitro antiproliferative and anti-HIV activity of new derivatives of 2-Piperazino-1,3-benzo[d]thiazoles | 1-Jan-2010 | AL SOUD, Ya; AL SA'DONI, Hh; Saber, Sow; AL SHANEEK, Rhm; AL MASOUDI, Na; Loddo, Roberta; LA COLLA, P. | ZEITSCHRIFT FÜR NATURFORSCHUNG. B, A JOURNAL OF CHEMICAL SCIENCES | - |
| Protective properties of non-nucleoside reverse transcriptase inhibitor (MC1220) incorporated into liposome against intravaginal challenge of Rhesus Macaques with RT-SHIV | 1-Jan-2010 | Caron, M; Besson, G; Etenna, Sl; MINTSA NDONG, A; Mourtas, S; Radaelli, A; Morghen, Cd; Loddo, Roberta; LA COLLA, P; Antimisiaris, Sg; Kazanji, M. | VIROLOGY | - |
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