Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives
2015-01-01 Briguglio, I; Loddo, Roberta; Laurini, E; Fermeglia, M; Piras, S; Corona, P; Giunchedi, P; Gavini, E; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; LA COLLA, Paolo; Pricl, S; Carta, A.
Synthesis, antimicrobial and pharmacological evalutation of thiourea-derivatives of 4H-1,2,4-triazole
2015-01-01 Bielenica, A; Kedzierska, E; Fidecka, S; Maluszynska, H; Miroslaw, B; Koziol, A. E.; Stefanska, J; Madeddu, Silvia; Giliberti, Gabriele; Sanna, Giuseppina; Struga, M.
Synthesis, cytotoxicity and antimicrobial activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety
2015-01-01 Bielenica, Anna; Stefanska, Joanna; Stepien, Karolina; Napiorkowska, Agnieszka; Augustynowicz Kopec, Ewa; Sanna, Giuseppina; Madeddu, Silvia; Boi, Stefano; Giliberti, Gabriele; Wrzosek, Malgorzata; Struga, Marta
Synthesis, antimicrobial and cytotoxic activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety
2015-01-01 A., Bielenica; J., Stefańska; K., Stępień; A., Napiórkowska; E., Augustynowicz Kopeć; Sanna, Giuseppina; Madeddu, S; S., Boi; Giliberti, Gabriele; M., Struga
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agents
2015-01-01 Spallarossa, Andrea; Caneva, Chiara; Caviglia, Matteo; Alfei, Silvana; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Brindisi, Margherita; Zisterer, Daniela M.; Bright, Sandra A.; Williams, Clive D.; Crespan, Emmanuele; Maga, Giovanni; Sanna, Giuseppina; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta
N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents
2015-01-01 Fioravanti, R; Desideri, N; Biava, M; Droghini, P; Atzori, Em; Ibba, Cristina; Collu, Gabriella; Sanna, Giuseppina; Delogu, Ilenia; Loddo, Roberta
Antimicrobial and anti-biofilm activity of thiourea derivatives incorporating 2-aminothiazole scaffold
2015-01-01 Stefanska, J; Nowicka, G; Struga, M; Szulczyk, D; Koziol, Ae; Augustynowicz Kopec, E; Napiorkowska, A; Bielenica, A; Filipowski, W; Filipowska, A; Drzewiecka, A; Giliberti, Gabriele; Madeddu, S; Boi, S; La Colla, P; Sanna, Giuseppina
Isolation and anticancer, anthelminthic, and antiviral (HIV) activity of acylphloroglucinols, and regioselective synthesis of empetrifranzinans from Hypericum roeperianum
2015-01-01 Fobofou, Sat; Franke, K; Sanna, Giuseppina; Porzel, A; Bullita, Enrica; LA COLLA, Paolo; Wessjohann, La
Synthesis, antimicrobial and pharmacological evaluation of thioureaderivatives of 4H-1,2,4-triazole
2015-01-01 Bielenica, A; Kedzierska, E; Fidecka, S; Maluszynska, A; Miroslaw, B; Koziol, Ae; Stefanska, J; Madeddu, Silvia; Giliberti, Gabriele; Sanna, Giuseppina; Struga, M.
Antiviral properties from plants of the Mediterranean flora
2015-01-01 Sanna, Giuseppina; Farci, P; Busonera, B; Murgia, G; La Colla, P; Giliberti, Gabriele
Antiviral activity of some aromatic and medicinal plants against RNA virus: preliminary study
2015-01-01 Madeddu, Silvia; Sanna, Giuseppina; Giliberti, Gabriele; Falconieri, Danilo; Porcedda, Silvia; Piras, Alessandra
Limonoids from Melia azedarach fruits as inhibitors of flaviviruses and mycobacterium tubercolosis
2015-01-01 Sanna, Giuseppina; Madeddu, Silvia; Giliberti, Gabriele; Ntalli, Nikoletta G.; Cottiglia, Filippo; DE LOGU, Alessandro; Agus, Emanuela; Caboni, Pierluigi
Synthesis of some new 2-amino-6-thiocyanato benzothiazole derivatives bearing 2,4-thiazolidinediones and screening of their in vitro antimicrobial, antitubercular and antiviral activities
2015-01-01 Faiyazalam, M; Saiyad, S; Navin B., P; Sanna, Giuseppina; B., Busonera; P., La Colla; Dhanji, P. R.
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents
2014-01-01 Tonelli, M; Novelli, F; Tasso, B; Vazzana, I; Sparatore, A; Boido, V; Sparatore, F; La Colla, P; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, B; Farci, P; Ibba, Cristina; Loddo, Roberta
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines
2014-01-01 Loddo, Roberta; Briguglio, I; Corona, P; Piras, S; Loriga, M; Paglietti, G; Carta, A; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, P; La Colla, P.
Synthesis of novel fluoro analogues of MKC442 as microbicides
2014-01-01 Loksha, Ym; Pedersen, Eb; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Giliberti, Gabriele; La Colla, P.
Synthesis and biological evaluation of N-substituted polycyclic imides derivatives
2013-01-01 Bielenica, A; Struga, M; Mirosław, B; Kozioł, Ae; Kossakowski, J; Sanna, Giuseppina; La Colla, P; Giliberti, Gabriele
Structural and antiviral studies of dipetalactone and its methyl derivative
2013-01-01 Drzewiecka, A; Koziol, Ae; Borowski, P; Sanna, Giuseppina; Giliberti, Gabriele; La Colla, P; Zawadowski, T; Struga, M.
Erratum to: Syntheses and in vitro biological screening of 1-aryl-10 H-[1,2,4]triazolo[3′,4′:3,4][1,2,4]triazino[5,6-b]indoles
2013-01-01 Upadhyay, K; Manvar, A; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A; Giliberti, Gabriele; Secci, B; Busonera, B; Sanna, Giuseppina; Loddo, Roberta; La Colla, P.
Cytotoxic phloroglucinols from the leaves of Myrtus communis
2012-01-01 Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina
Disubstituted thiourea derivatives and their activity on CNS: Synthesis and biological evaluation
2012-01-01 Stefanska, J; Szulczyk, D; Koziol, Ae; Miroslaw, B; Kedzierska, E; Fidecka, S; Busonera, B; Sanna, Giuseppina; Giliberti, Gabriele; La Colla, P; Struga, M.
Potent and Selective Activity of Daphnane Diterpens against HIV-1, HIV-2 and Coxsackievirus
2012-01-01 Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; La Colla, P.
A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220
2012-01-01 Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, R; La Colla, P.
A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220
2012-01-01 Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, Roberta; La Colla, P.
5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4
2012-01-01 Vitale, G; Corona, P; Loriga, M; Carta, M; Paglietti, G; Giliberti, Gabriele; Sanna, Giuseppina; Farci, P; Marongiu, Me; La Colla, P.
Phenyl-benzotriazoles: new potent and selective inhibitors of Respiratory Syncytial Virus and Hantaviruses
2011-01-01 Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; Farci, P; Marongiu M., E; La Colla, P.
Bioguided-isolation of cytotoxic phloroglucinols from the leaves of myrtus communis l.
2011-01-01 Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, P; Aicha, O; Sanna, Giuseppina
Phenyl-benzotriazoles: new potent and selective inhibitors of Respiratory Syncytial and Hanta viruses
2011-01-01 Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; Farci, P; Marongiu, Me; La Colla, P.
(Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity
2010-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; La Colla, P; Collu, G; Sanna, Giuseppina; Loddo, R.
1,2-benzisothiazol-3(2h)-one benzenesulfonamides targeting the hiv nucleocapsid proteins are potential microbicide candidates for the prevention of mucosal hiv transmission/acquisition
2010-01-01 Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; Giliberti, Gabriele; Marongiu, E.; Loddo, Roberta; La Colla, P.
Antiviral activity of benzimidazole derivatives. II. Antiviral activity of 2-phenylbenzimidazole derivatives
2010-01-01 Tonelli, M; Simone, M; Tasso, B; Novelli, F; Boido, V; Sparatore, F; Paglietti, G; Pricl, S; Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Ibba, Cristina; Sanna, Giuseppina; Loddo, Roberta; La Colla, P.
1,2-benzisothiazol-3(2H)-one benzenesulfonamides as new microbicide candidates for prevention of mucosal HIV infections
2009-01-01 Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; Sanna, Giuseppina; Secci, B; Marongiu, E; Loddo, Roberta; La Colla, P.
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Schenone, S; Bruno, O; Borassi, A; LA COLLA, P; Pezzullo, M; Sanna, Giuseppina; Collu, Gabriella; Secci, Barbara; Loddo, Roberta
N-acylated and N,N’-diacylated imidazolidine-2-thione derivatives and N,N’-diacylated tetrahydropyrimidine-2(1H)-thione analogues: synthesis and antiproliferative activity
2009-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Rosano, C; LA COLLA, P; Sanna, Giuseppina; Busonera, B; Loddo, Roberta
Synthesis of novel uracil non-nucleoside derivatives as potential reverse transcriptase inhibitors of HIV-1
2009-01-01 El Brollosy, Nr; Al Deeb, Oa; El Emam, Aa; Pedersen, Eb; La Colla, P; Collu, G; Sanna, Giuseppina; Loddo, Roberta
Synthesis, pharmacological and antiviral activity of 1,3-thiazepine derivatives
2009-01-01 Struga, M; Kossakowski, J; Koziol, Ae; Kedzierska, E; Fidecka, S; LA COLLA, P; Ibba, Cristina; Collu, G; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta
Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters
2009-01-01 Romanowska, J; SZYMANSKA MICHALAK, A; Boryski, J; Stawinski, J; Kraszewski, A; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Secci, Barbara; LA COLLA, P.
Anti-retroviral activity of novel 1,2-benzisothiazol-3(2H)-one benzenesulfonamides targeting HIV nucleocapsid (NC) proteins
2009-01-01 Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; La Colla, P.
Results on different formulations of an NNRTI candidate (MC 1220) for application as topical microbicide
2009-01-01 Blois, SYLVAIN SERGE DANIEL; Marongiu, E; Sanna, Giuseppina; Collu, G; Secci, B; Giliberti, Gabriele; Loddo, Roberta; Pedersen, E; De Giuli Morghen, C; Stahl Hennig, C; La Colla, P.
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
2009-01-01 Spallarossa, A; Cesarini, S; Ranise, A; Bruno, O; Schenone, S; LA COLLA, P; Collu, Gabriella; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Bruno, O; LA COLLA, P; Casula, L; Collu, Gabriella; Sanna, Giuseppina; Loddo, Roberta
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents.
2008-01-01 Spallarossa, A; Cesarini, S; Rotolo, C; Fossa, P; Mosti, L; Ranise, A; Sanna, Giuseppina; Collu, G; Secci, B; Busonera, B; La Colla, P; Loddo, R.
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates
2008-01-01 Cesarini, S; Spallarossa, A; Ranise, A; Fossa, P; LA COLLA, P; Sanna, Giuseppina; Collu, G; Loddo, Roberta
Polymers as potent inhibitors of HIV-1. Europrise, Rational Design of HIV
2008-01-01 Secci, B; Sanna, Giuseppina; Collu, G; La Colla, P; Loddo, R.
Synthesis and antiviral activity of new dimeric inhibitors against HIV-1
2008-01-01 Danel, K; Larsen, Lm; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta
Synthesis and antiviral evaluation of 6-(trifluoromethylbenzyl) and 6-(fluorobenzyl) analogues of HIV drugs Emivirine and GCA-186
2008-01-01 EL BROLLOSY, Nr; Sørensen, Er; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta
In vitro evaluation of the anti-HIV-1 activity of Liposomes and gel ingredients
2008-01-01 Loddo, Roberta; Sanna, Giuseppina; Collu, G; Busonera, B; Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; La Colla, P.
In vitro evaluation of the anti-HIV-1 activity of liposomes and gel ingredients
2006-01-01 Loddo, Roberta; Sanna, Giuseppina; Collu, G; Busonera, B; Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; La Colla, P.
Hindered nucleoside analogs as inhibitors of HCV RNA-dependent RNA polymerase: evolving vistas
2006-01-01 Manfredini, S; Angusti, A; Ciliberti, N; Durini, E; Vertuani, S; Buzzoni, L; Coslanich, A; Fermeglia, M; Ferrone, M; PANENI M., S; Pricl, S; LA COLLA, P; Sanna, Giuseppina; Cadeddu, A; Mura, M; Loddo, Roberta
Extraction of Juniperus communis L. ssp. nana Willd. essential oil by supercritical carbon dioxide
2006-01-01 Marongiu, B; Porcedda, Silvia; Piras, Alessandra; Sanna, Giuseppina; Mureddu, M; Loddo, Roberta
Title | Issue Date | Author(s) | Journal | Publisher |
---|---|---|---|---|
Synthesis, cytotoxicity and antiviral evaluation of new series of imidazo[4,5-g]quinoline and pyrido[2,3-g]quinoxalinone derivatives | 1-Jan-2015 | Briguglio, I; Loddo, Roberta; Laurini, E; Fermeglia, M; Piras, S; Corona, P; Giunchedi, P; Gavini, E; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, Pamela; LA COLLA, Paolo; Pricl, S; Carta, A. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis, antimicrobial and pharmacological evalutation of thiourea-derivatives of 4H-1,2,4-triazole | 1-Jan-2015 | Bielenica, A; Kedzierska, E; Fidecka, S; Maluszynska, H; Miroslaw, B; Koziol, A. E.; Stefanska, J; Madeddu, Silvia; Giliberti, Gabriele; Sanna, Giuseppina; Struga, M. | LETTERS IN DRUG DESIGN & DISCOVERY | - |
Synthesis, cytotoxicity and antimicrobial activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety | 1-Jan-2015 | Bielenica, Anna; Stefanska, Joanna; Stepien, Karolina; Napiorkowska, Agnieszka; Augustynowicz Kopec, Ewa; Sanna, Giuseppina; Madeddu, Silvia; Boi, Stefano; Giliberti, Gabriele; Wrzosek, Malgorzata; Struga, Marta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis, antimicrobial and cytotoxic activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moiety | 1-Jan-2015 | A., Bielenica; J., Stefańska; K., Stępień; A., Napiórkowska; E., Augustynowicz Kopeć; Sanna, Giuseppina; Madeddu, S; S., Boi; Giliberti, Gabriele; M., Struga | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agents | 1-Jan-2015 | Spallarossa, Andrea; Caneva, Chiara; Caviglia, Matteo; Alfei, Silvana; Butini, Stefania; Campiani, Giuseppe; Gemma, Sandra; Brindisi, Margherita; Zisterer, Daniela M.; Bright, Sandra A.; Williams, Clive D.; Crespan, Emmanuele; Maga, Giovanni; Sanna, Giuseppina; Delogu, Ilenia; Collu, Gabriella; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents | 1-Jan-2015 | Fioravanti, R; Desideri, N; Biava, M; Droghini, P; Atzori, Em; Ibba, Cristina; Collu, Gabriella; Sanna, Giuseppina; Delogu, Ilenia; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | - |
Antimicrobial and anti-biofilm activity of thiourea derivatives incorporating 2-aminothiazole scaffold | 1-Jan-2015 | Stefanska, J; Nowicka, G; Struga, M; Szulczyk, D; Koziol, Ae; Augustynowicz Kopec, E; Napiorkowska, A; Bielenica, A; Filipowski, W; Filipowska, A; Drzewiecka, A; Giliberti, Gabriele; Madeddu, S; Boi, S; La Colla, P; Sanna, Giuseppina | CHEMICAL & PHARMACEUTICAL BULLETIN | - |
Isolation and anticancer, anthelminthic, and antiviral (HIV) activity of acylphloroglucinols, and regioselective synthesis of empetrifranzinans from Hypericum roeperianum | 1-Jan-2015 | Fobofou, Sat; Franke, K; Sanna, Giuseppina; Porzel, A; Bullita, Enrica; LA COLLA, Paolo; Wessjohann, La | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Synthesis, antimicrobial and pharmacological evaluation of thioureaderivatives of 4H-1,2,4-triazole | 1-Jan-2015 | Bielenica, A; Kedzierska, E; Fidecka, S; Maluszynska, A; Miroslaw, B; Koziol, Ae; Stefanska, J; Madeddu, Silvia; Giliberti, Gabriele; Sanna, Giuseppina; Struga, M. | LETTERS IN DRUG DESIGN & DISCOVERY | - |
Antiviral properties from plants of the Mediterranean flora | 1-Jan-2015 | Sanna, Giuseppina; Farci, P; Busonera, B; Murgia, G; La Colla, P; Giliberti, Gabriele | NATURAL PRODUCT RESEARCH | - |
Antiviral activity of some aromatic and medicinal plants against RNA virus: preliminary study | 1-Jan-2015 | Madeddu, Silvia; Sanna, Giuseppina; Giliberti, Gabriele; Falconieri, Danilo; Porcedda, Silvia; Piras, Alessandra | - | - |
Limonoids from Melia azedarach fruits as inhibitors of flaviviruses and mycobacterium tubercolosis | 1-Jan-2015 | Sanna, Giuseppina; Madeddu, Silvia; Giliberti, Gabriele; Ntalli, Nikoletta G.; Cottiglia, Filippo; DE LOGU, Alessandro; Agus, Emanuela; Caboni, Pierluigi | PLOS ONE | - |
Synthesis of some new 2-amino-6-thiocyanato benzothiazole derivatives bearing 2,4-thiazolidinediones and screening of their in vitro antimicrobial, antitubercular and antiviral activities | 1-Jan-2015 | Faiyazalam, M; Saiyad, S; Navin B., P; Sanna, Giuseppina; B., Busonera; P., La Colla; Dhanji, P. R. | MEDICINAL CHEMISTRY RESEARCH | - |
Antiviral activity of benzimidazole derivatives. III. Novel anti-CVB-5, anti-RSV and anti-Sb-1 agents | 1-Jan-2014 | Tonelli, M; Novelli, F; Tasso, B; Vazzana, I; Sparatore, A; Boido, V; Sparatore, F; La Colla, P; Sanna, Giuseppina; Giliberti, Gabriele; Busonera, B; Farci, P; Ibba, Cristina; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Synthesis and antiviral activity of new phenylimidazopyridines and N-benzylidenequinolinamines derived by molecular simplification of phenylimidazo[4,5-g]quinolines | 1-Jan-2014 | Loddo, Roberta; Briguglio, I; Corona, P; Piras, S; Loriga, M; Paglietti, G; Carta, A; Sanna, Giuseppina; Giliberti, Gabriele; Ibba, Cristina; Farci, P; La Colla, P. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis of novel fluoro analogues of MKC442 as microbicides | 1-Jan-2014 | Loksha, Ym; Pedersen, Eb; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Giliberti, Gabriele; La Colla, P. | JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis and biological evaluation of N-substituted polycyclic imides derivatives | 1-Jan-2013 | Bielenica, A; Struga, M; Mirosław, B; Kozioł, Ae; Kossakowski, J; Sanna, Giuseppina; La Colla, P; Giliberti, Gabriele | ACTA POLONIAE PHARMACEUTICA | - |
Structural and antiviral studies of dipetalactone and its methyl derivative | 1-Jan-2013 | Drzewiecka, A; Koziol, Ae; Borowski, P; Sanna, Giuseppina; Giliberti, Gabriele; La Colla, P; Zawadowski, T; Struga, M. | JOURNAL OF MOLECULAR STRUCTURE | - |
Erratum to: Syntheses and in vitro biological screening of 1-aryl-10 H-[1,2,4]triazolo[3′,4′:3,4][1,2,4]triazino[5,6-b]indoles | 1-Jan-2013 | Upadhyay, K; Manvar, A; Virsodiya, V; Trivedi, J; Chaniyara, R; Shah, A; Giliberti, Gabriele; Secci, B; Busonera, B; Sanna, Giuseppina; Loddo, Roberta; La Colla, P. | MEDICINAL CHEMISTRY RESEARCH | - |
Cytotoxic phloroglucinols from the leaves of Myrtus communis | 1-Jan-2012 | Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, Pamela; Ouhtit, A; Sanna, Giuseppina | JOURNAL OF NATURAL PRODUCTS | - |
Disubstituted thiourea derivatives and their activity on CNS: Synthesis and biological evaluation | 1-Jan-2012 | Stefanska, J; Szulczyk, D; Koziol, Ae; Miroslaw, B; Kedzierska, E; Fidecka, S; Busonera, B; Sanna, Giuseppina; Giliberti, Gabriele; La Colla, P; Struga, M. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Potent and Selective Activity of Daphnane Diterpens against HIV-1, HIV-2 and Coxsackievirus | 1-Jan-2012 | Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; La Colla, P. | - | - |
A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220 | 1-Jan-2012 | Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, R; La Colla, P. | - | - |
A Computationally-Based Explanation for the Knocking Out Activity of the Microbicide MC1220 | 1-Jan-2012 | Giliberti, Gabriele; Asthana, S; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Busonera, B; Loddo, Roberta; La Colla, P. | - | - |
5-Acetyl-2-arylbenzimidazoles as antiviral agents. Part 4 | 1-Jan-2012 | Vitale, G; Corona, P; Loriga, M; Carta, M; Paglietti, G; Giliberti, Gabriele; Sanna, Giuseppina; Farci, P; Marongiu, Me; La Colla, P. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Phenyl-benzotriazoles: new potent and selective inhibitors of Respiratory Syncytial Virus and Hantaviruses | 1-Jan-2011 | Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; Farci, P; Marongiu M., E; La Colla, P. | - | - |
Bioguided-isolation of cytotoxic phloroglucinols from the leaves of myrtus communis l. | 1-Jan-2011 | Cottiglia, Filippo; Casu, Laura; Leonti, Marco; Caboni, Pierluigi; Floris, Costantino; Busonera, B; Farci, P; Aicha, O; Sanna, Giuseppina | - | - |
Phenyl-benzotriazoles: new potent and selective inhibitors of Respiratory Syncytial and Hanta viruses | 1-Jan-2011 | Sanna, Giuseppina; Busonera, B; Giliberti, Gabriele; Farci, P; Marongiu, Me; La Colla, P. | - | - |
(Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity | 1-Jan-2010 | Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; La Colla, P; Collu, G; Sanna, Giuseppina; Loddo, R. | MEDICINAL CHEMISTRY RESEARCH | - |
1,2-benzisothiazol-3(2h)-one benzenesulfonamides targeting the hiv nucleocapsid proteins are potential microbicide candidates for the prevention of mucosal hiv transmission/acquisition | 1-Jan-2010 | Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; Giliberti, Gabriele; Marongiu, E.; Loddo, Roberta; La Colla, P. | - | - |
Antiviral activity of benzimidazole derivatives. II. Antiviral activity of 2-phenylbenzimidazole derivatives | 1-Jan-2010 | Tonelli, M; Simone, M; Tasso, B; Novelli, F; Boido, V; Sparatore, F; Paglietti, G; Pricl, S; Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Ibba, Cristina; Sanna, Giuseppina; Loddo, Roberta; La Colla, P. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
1,2-benzisothiazol-3(2H)-one benzenesulfonamides as new microbicide candidates for prevention of mucosal HIV infections | 1-Jan-2009 | Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; Sanna, Giuseppina; Secci, B; Marongiu, E; Loddo, Roberta; La Colla, P. | - | - |
Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors | 1-Jan-2009 | Spallarossa, A; Cesarini, S; Ranise, A; Schenone, S; Bruno, O; Borassi, A; LA COLLA, P; Pezzullo, M; Sanna, Giuseppina; Collu, Gabriella; Secci, Barbara; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
N-acylated and N,N’-diacylated imidazolidine-2-thione derivatives and N,N’-diacylated tetrahydropyrimidine-2(1H)-thione analogues: synthesis and antiproliferative activity | 1-Jan-2009 | Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Rosano, C; LA COLLA, P; Sanna, Giuseppina; Busonera, B; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Synthesis of novel uracil non-nucleoside derivatives as potential reverse transcriptase inhibitors of HIV-1 | 1-Jan-2009 | El Brollosy, Nr; Al Deeb, Oa; El Emam, Aa; Pedersen, Eb; La Colla, P; Collu, G; Sanna, Giuseppina; Loddo, Roberta | ARCHIV DER PHARMAZIE | - |
Synthesis, pharmacological and antiviral activity of 1,3-thiazepine derivatives | 1-Jan-2009 | Struga, M; Kossakowski, J; Koziol, Ae; Kedzierska, E; Fidecka, S; LA COLLA, P; Ibba, Cristina; Collu, G; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Aryl nucleoside H-phosphonates. Part 16: synthesis and anti-HIV-1 activity of di-aryl nucleoside phosphotriesters | 1-Jan-2009 | Romanowska, J; SZYMANSKA MICHALAK, A; Boryski, J; Stawinski, J; Kraszewski, A; Loddo, Roberta; Sanna, Giuseppina; Collu, G; Secci, Barbara; LA COLLA, P. | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Anti-retroviral activity of novel 1,2-benzisothiazol-3(2H)-one benzenesulfonamides targeting HIV nucleocapsid (NC) proteins | 1-Jan-2009 | Giliberti, Gabriele; Blois, SYLVAIN SERGE DANIEL; Sanna, Giuseppina; Secci, B; La Colla, P. | - | - |
Results on different formulations of an NNRTI candidate (MC 1220) for application as topical microbicide | 1-Jan-2009 | Blois, SYLVAIN SERGE DANIEL; Marongiu, E; Sanna, Giuseppina; Collu, G; Secci, B; Giliberti, Gabriele; Loddo, Roberta; Pedersen, E; De Giuli Morghen, C; Stahl Hennig, C; La Colla, P. | - | - |
Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors | 1-Jan-2009 | Spallarossa, A; Cesarini, S; Ranise, A; Bruno, O; Schenone, S; LA COLLA, P; Collu, Gabriella; Sanna, Giuseppina; Secci, Barbara; Loddo, Roberta | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | - |
Parallel one-pot synthesis and structure-activity relationship study of symmetric formimidoester disulfides as a novel class of potent non-nucleoside HIV-1 reverse transcriptase inhibitors | 1-Jan-2008 | Cesarini, S; Spallarossa, A; Ranise, A; Schenone, S; Bruno, O; LA COLLA, P; Casula, L; Collu, Gabriella; Sanna, Giuseppina; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents. | 1-Jan-2008 | Spallarossa, A; Cesarini, S; Rotolo, C; Fossa, P; Mosti, L; Ranise, A; Sanna, Giuseppina; Collu, G; Secci, B; Busonera, B; La Colla, P; Loddo, R. | - | - |
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates | 1-Jan-2008 | Cesarini, S; Spallarossa, A; Ranise, A; Fossa, P; LA COLLA, P; Sanna, Giuseppina; Collu, G; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Polymers as potent inhibitors of HIV-1. Europrise, Rational Design of HIV | 1-Jan-2008 | Secci, B; Sanna, Giuseppina; Collu, G; La Colla, P; Loddo, R. | - | - |
Synthesis and antiviral activity of new dimeric inhibitors against HIV-1 | 1-Jan-2008 | Danel, K; Larsen, Lm; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta | BIOORGANIC & MEDICINAL CHEMISTRY | - |
Synthesis and antiviral evaluation of 6-(trifluoromethylbenzyl) and 6-(fluorobenzyl) analogues of HIV drugs Emivirine and GCA-186 | 1-Jan-2008 | EL BROLLOSY, Nr; Sørensen, Er; Pedersen, Eb; Sanna, Giuseppina; LA COLLA, P; Loddo, Roberta | ARCHIV DER PHARMAZIE | - |
In vitro evaluation of the anti-HIV-1 activity of Liposomes and gel ingredients | 1-Jan-2008 | Loddo, Roberta; Sanna, Giuseppina; Collu, G; Busonera, B; Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; La Colla, P. | - | - |
In vitro evaluation of the anti-HIV-1 activity of liposomes and gel ingredients | 1-Jan-2006 | Loddo, Roberta; Sanna, Giuseppina; Collu, G; Busonera, B; Blois, SYLVAIN SERGE DANIEL; Giliberti, Gabriele; La Colla, P. | - | - |
Hindered nucleoside analogs as inhibitors of HCV RNA-dependent RNA polymerase: evolving vistas | 1-Jan-2006 | Manfredini, S; Angusti, A; Ciliberti, N; Durini, E; Vertuani, S; Buzzoni, L; Coslanich, A; Fermeglia, M; Ferrone, M; PANENI M., S; Pricl, S; LA COLLA, P; Sanna, Giuseppina; Cadeddu, A; Mura, M; Loddo, Roberta | - | - |
Extraction of Juniperus communis L. ssp. nana Willd. essential oil by supercritical carbon dioxide | 1-Jan-2006 | Marongiu, B; Porcedda, Silvia; Piras, Alessandra; Sanna, Giuseppina; Mureddu, M; Loddo, Roberta | FLAVOUR AND FRAGRANCE JOURNAL | - |
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