Dmt-Tic-OH a highly selective and potent delta-opioid dipeptide receptor antagonist after systemic administration in the mouse
1996-01-01 Capasso, A.; Guerrini, R.; Balboni, Gianfranco; Sorrentino, R.; Temussi, P.; Lazarus, L. H.; Bryant, S. D.; Salvadori, S.
Solution and Solid-State Structure of the diketopiperazine of tyrosyl-tetrahydroisoquinoline-3-carboxylic Acid
1995-01-01 Ciajolo, Mr; Balboni, Gianfranco; Picone, D; Salvadori, S; Tancredi, T; Temussi, Pa; Tuzi, A.
Acid Catalysis in the Formation of dioxopiperazines from Peptides containing tetrahydroisoquinoline-3-carboxylic acid at Position 2
1995-01-01 Capasso, S; Sica, F; Mazzarella, L; Balboni, Gianfranco; Guerrini, R; Salvadori, S.
Delta opioidmimetic antagonists: prototypes for designing a new generation of ultraselective opioid peptides
1995-01-01 Salvadori, S.; Attila, M.; Balboni, Gianfranco; Bianchi, C.; Bryant, S. D.; Crescenzi, O.; Guerrini, R.; Picone, D.; Tancredi, T.; Tamussi, P. A.
Single diastereomeric desaminotyrosylalanyl tetra- and heptapeptides with Opioid Antagonist Activity
1995-01-01 Balboni, Gianfranco; Salvadori, S; D'Angeli, F; Marchetti, P; Lazarus, Lh; Bryant, Sd; Bianchi, C.
Conformational analysis of potent and very selective delta opioid dipeptide antagonists
1995-01-01 Amodeo, P.; Balboni, Gianfranco; Crescenzi, O.; Guerrini, R.; Picone, D.; Salvadori, S.; Tancredi, T.; Temussi, P. A.
Synthesis and Opioid Activity of tyrosine sulfate containing dermorphin and Deltorphin Peptides
1995-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Scaranari, V; Borea, Pa; Tomatis, A.
Structure-activity ralationships of cyclic and linear peptide T analogues
1993-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Scaranari, V; Spisani, S; Reali, E; Traniello, S; Tomatis, R.
Synthesis and receptor binding analysis of dermorphin hepta-, hexa- and pentapeptide analogues. Evidence for one- and two-side binding models for the mu-opioid receptor
1993-01-01 Attila, M; Salvadori, S; Balboni, Gianfranco; Bryant, Sd; Lazarus, Lh
Phe3-substituted analogues of deltorphin C. Spatial conformation and topography of the aromatic ring in peptide recognition by delta opioid receptors
1993-01-01 Salvadori, S; Bryant, Sd; Bianchi, C; Balboni, Gianfranco; Scaranari, V; Attila, M; Lazarus, Lh
2-bromoamides as synthons for pseudopeptides containing aminodicarboxy units
1993-01-01 D'Angeli, F; Marchetti, P; Salvadori, S; Balboni, Gianfranco
Linear oligopeptides. 252. alpha,beta-dehydro-amino acid residues in the design of peptide structures - molecular and crystal-stuctures of 2 folded dehydro peptides
1992-01-01 Busetti, V; Crisma, M; Toniolo, C; Salvadori, S; Balboni, Gianfranco
Alterations in vasoactive intestinal polypeptide-related peptides after pentylenetetrazole-induced seizures in rat brain
1992-01-01 Romualdi, P; Lesa, G; Donatini, A; Balboni, Gianfranco; Tomatis, R; Ferri, S.
Stereospecificity of amino acid side chains in deltorphin defines binding to opioid receptors
1992-01-01 Lazarus, Lh; Salvadori, S; Balboni, Gianfranco; Tomatis, R; Wilson, We
On the degradation of the deltorphin peptides by plasma and brain homogenate
1991-01-01 Marastoni, M; Tomatis, R; Balboni, Gianfranco; Salvadori, S; Lazarus, Lh
Studies on the anti-phospholipase A2 and anti-inflammatory activities of a synthetic nonapeptide from uteroglobin
1991-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Scaranari, V; Santagada, V; Romualdi, P; Ferri, S; Tomatis, R.
New insights on the mu/delta selectivity of opioid peptides: conformational analysis of deltorphin analogues
1991-01-01 Tancredi, T; Temussi, Pa; Picone, D; Amodeo, P; Tomatis, R; Salvadori, S; Marastoni, M; Santagada, V; Balboni, Gianfranco
Synthesis and structure-activity relationships of deltorphin analogues
1991-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Borea, Pa; Morari, M; Tomatis, R.
Chemotactic response of human monocytes to pentapeptide analog derived from immunodeficiency virus protein gp 120
1990-01-01 Spisani, S; Gavioli, R; Giuliani, Al; Cavalletti, T; Marastoni, M; Balboni, Gianfranco; Salvadori, S; Tomatis, R; Traniello, S.
Opioid peptides. Synthesis and biological properties of dermorphin related hexapeptides
1990-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Borea, P; Tomatis, R.
New features of the delta opioid receptor: conformationalproperties of deltorphin I analogues
1990-01-01 Balboni, Gianfranco; Marastoni, M; Picone, D; Salvadori, S; Tancredi, T; Temussi, Pa; Tomatis, R.
Synthesis, metabolic stability and chemotactic activity of peptide T and its analogues
1990-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Spisani, S; Gavioli, R; Traniello, S; Tomatis, R.
NMR studies of a series of dehydrodermorphins
1989-01-01 CASTIGLIONE MORELLI, Ma; Saviano, G; Temussi, Pa; Balboni, Gianfranco; Salvadori, S; Tomatis, R.
Opioid peptides. Synthesis and binding properties of dermorphin related heptapeptides
1989-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Borea, P; Tomatis, R.
Conformational properties of deltorphin: new features of the delta-opioid receptor
1989-01-01 Temussi, Pa; Picone, D; Tancredi, T; Tomatis, R; Salvadori, S; Marastoni, M; Balboni, Gianfranco
Structure-activity relationships of peptide T-related pentapeptides
1989-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Spisani, S; Gavioli, R; Traniello, S; Tomatis, R.
Opioid peptides. Partially modified retro-inverso dermorphin analogues. XIII
1989-01-01 Marastoni, M; Balboni, Gianfranco; Tomatis, R; Salvadori, S; Borea, Pa; Uccelli, L.
Synthesis and activity of dermorphin-growth hormone releasing factor hybrid peptides
1989-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Borea, Pa; Tomatis, R.
Structure-activity relatioships of tetrapeptides related to dermorphin: a 500-MHz 1H-nmr study
1988-01-01 CASTIGLIONE MORELLI, Ma; Tancredi, T; Trivellone, E; Balboni, Gianfranco; Marastoni, M; Salvadori, S; Tomatis, R; Temussi, Pa
Opioid agonists and antagonists - Peptides containing N-terminal allyl groups and or a thiomethylene linkage in place of a peptide-bond
1988-01-01 Balboni, Gianfranco; Salvadori, S; Marastoni, M; Tomatis, R; Borea, Pa; Bianchi, C.
Synthesis and activity profiles of new dermorphin-(1-4) peptide analogues
1987-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Borea, Pa; Marzola, G; Tomatis, R.
Opioid peptides. Synthesis and binding assays of desamino-Tyr1 dermorphin analogues. XII
1987-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Tomatis, R; Borea, Pa
Dehydro-dermorphins. II. Synthesis and biological activity of unsatured dermorphin hexa and heptapeptides
1986-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Marzila, G; Tomatis, R.
Synthesis and biological activity of carboxyl terminally extended ermorphins
1986-01-01 Marastoni, M; Salvadori, S; Balboni, Gianfranco; Marzola, G; DEGLI UBERTI, Ec; Tomatis, R.
Synthesis and opioid activity of dermorphin tetrapeptides beearing D-methionine S-oxide at position 2
1986-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Sarto, Gp; Tomatis, R.
Dehydro-dermorphins. I. Influence of the stereo-orientation of aromatic groups in dermorphin-(1-5)-peptides to opioid activity
1986-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Marzola, G; Tomatis, R.
Dehydro-dermorphins. III. Circular dichroism investigation of conformation in solution
1986-01-01 Pieroni, O; Fissi, A; Salvadori, S; Balboni, Gianfranco; Tomatis, R.
Synthesis and opioid activity of partially retro-inverso analogs of dermorphin
1985-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Sarto, G; Tomatis, R.
Synthesis and pharmacological activity of partially modified retro-inverso dermorphin tetrapeptides
1985-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Sarto, Gp; Tomatis, R.
Opioid peptides. VIII. Synthesis and preliminary biological activity of [D-Phe3]- or [alpha,beta-dehydro-Phe3]dermorphin tetrapeptides
1985-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Tomatis, R.
Structure-activity relatioships of dermorphin tetrapeptides carrying a ketomethylene linkage
1985-01-01 Marastoni, M; Balboni, Gianfranco; Salvadori, S; Sarto, Gp; Tomatis, R.
Synthetic tetrapeptides related to dermorphin: potent long lasting analgesic action following subcutaneous administration
1985-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; DEGLI UBERTI, E; Tomatis, R.
Synthesis and opioid activity of [Sar4]dermorphin-tetrapeptide analogues
1984-01-01 Salvadori, S; Balboni, Gianfranco; Marastoni, M; Sarto, G; Tomatis, R.
Opioid peptides: Structure-activity relationships of dermorphin endothiotetrapeptides. VII
1984-01-01 Salvadori, S; Marastoni, M; Balboni, Gianfranco; Tomatis, R; Sarto, G.
Base-promoted reactions of alpha-halogeno-alkylanilides
1982-01-01 Cavicchioni, G; Scrimin, P; Veronese, Ac; Balboni, Gianfranco; D'Angeli, F.
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